Compile Data Set for Download or QSAR
maximum 50k data
Found 58 of ic50 data for polymerid = 49000526,50000019,50000150,50000462,50002350
LigandPNGBDBM50488134(CHEMBL2283229)
Affinity DataIC50:  73nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488117(CHEMBL2283230)
Affinity DataIC50:  91nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488133(CHEMBL2283231)
Affinity DataIC50:  110nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488132(CHEMBL2283321)
Affinity DataIC50:  130nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488131(CHEMBL2283322)
Affinity DataIC50:  140nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488142(CHEMBL2283232)
Affinity DataIC50:  150nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488139(CHEMBL2283323)
Affinity DataIC50:  200nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488140(CHEMBL2283221)
Affinity DataIC50:  240nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488130(CHEMBL2283208)
Affinity DataIC50:  280nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488116(CHEMBL2283209)
Affinity DataIC50:  300nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488136(CHEMBL2283222)
Affinity DataIC50:  320nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488123(CHEMBL2283223)
Affinity DataIC50:  370nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488122(CHEMBL2283224)
Affinity DataIC50:  460nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488119(CHEMBL2283210)
Affinity DataIC50:  560nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488120(CHEMBL2283225)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488121(CHEMBL2283226)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50255245(3-chloro-1-(4-hydroxyphenyl)propan-1-one | CHEMBL5...)
Affinity DataIC50:  3.99E+3nMAssay Description:Inhibition of GABA transaminase in rat brain by Kitz-Wilson plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50488118(CHEMBL2283227)
Affinity DataIC50:  4.96E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177407(1-(4-hydroxyphenyl)prop-2-en-1-one | 4-acryloylphe...)
Affinity DataIC50:  5.48E+3nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50488135(CHEMBL2283228)
Affinity DataIC50:  6.54E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488129(CHEMBL2283211)
Affinity DataIC50:  9.95E+3nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488128(CHEMBL2283212)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Mus musculus)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510591(CHEMBL4521189)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177412(4-(aminomethyl)phenol | 4-hydroxybenzylamine | CHE...)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177410(4-hydroxy-3-nitrobenzaldehyde | CHEMBL378361)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50488138(CHEMBL2283213)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50177411(4-formylphenol | 4-hydroxybenzaldehyde | CHEMBL141...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of GABA transaminase in rat brain by Kitz-Wilson plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177411(4-formylphenol | 4-hydroxybenzaldehyde | CHEMBL141...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50488141(CHEMBL2283214)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177405(3-methoxy-4-hydroxybenzaldehyde | 4-hydroxy-3-meth...)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50488127(CHEMBL2283215)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488137(CHEMBL2283216)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488115(CHEMBL2283217)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488126(CHEMBL2283218)
Affinity DataIC50:  2.59E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50488125(CHEMBL2283219)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Mus musculus)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataIC50:  3.97E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50118886(4-Amino-hex-5-enoic acid | CHEMBL89598 | US1018980...)
Affinity DataIC50:  4.12E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50488124(CHEMBL2283220)
Affinity DataIC50:  4.41E+4nMAssay Description:Inhibition of Rattus norvegicus (rat) brain gamma-amino butyrate aminotransferase using gamma-amino butyrate as substrate assessed as decrease in NAD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
Target4-aminobutyrate aminotransferase, mitochondrial(Mus musculus)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510593(CHEMBL4569177)
Affinity DataIC50:  5.14E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Mus musculus)
Jouf University

Curated by ChEMBL
LigandPNGBDBM50510592(CHEMBL4452708)
Affinity DataIC50:  5.81E+4nMAssay Description:Inhibition of GABA aminotransferase in mouse brain homogenates using GABA and alpha-ketoglutarate as substrates preincubated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177402(1-(4-hydroxy-phenyl)-propan-1-one | 1-(4-hydroxyph...)
Affinity DataIC50:  1.76E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177409((4-hydroxyphenyl)ethan-1-one | 1-(4-hydroxyphenyl)...)
Affinity DataIC50:  1.88E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177406(4-hydroxybenzaldehyde oxime | CHEMBL202611)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177408(4-(hydroxymethyl)phenol | 4-Hydroxybenzyl alcohol ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50139370(4-Methoxy-benzaldehyde | 4-methoxybenzaldehyde | C...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177404(4-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymet...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50145829(4-Aminobenzoesaeure | 4-aminobenzoic acid | CHEMBL...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM26194(4-Hydroxybenzoate, III | 4-hydroxybenzoic acid | C...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177413(4-hydroxy-3-methoxybenzaldehyde oxime | CHEMBL2024...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Huazhong University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50177403((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(4-(hydroxyme...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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