Report error Found 2274 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1D'
Affinity DataEC50: 5.01nMAssay Description:Agonist activity at human 5-HT1D receptor expressed in CHO cells assessed as stimulation of GTPgammaS binding by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human 5-HT1D receptor expressed in CHO cells assessed as stimulation of GTPgammaS binding by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Compound was tested for the inhibition of forskolin-stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptor in guinea pig substantia nigraMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Compound was tested for the inhibition of forskolin-stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptor in guinea pig substantia nigraMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0420nMAssay Description:Compound was tested for the inhibition of forskolin-stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptor in guinea pig substantia nigraMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.450nMAssay Description:Compound was tested for its ability inhibit forskolin-stimulated activity of adenylate cyclase coupled to human 5-HT 1D-beta receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Forskolin-stimulated adenylate cyclase activity against 5-hydroxytryptamine 1D receptor of rat substantia nigraMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Inhibition of Forskolin-stimulated adenylate cyclase activity against 5-hydroxytryptamine 1D receptor of guinea pig substantia nigraMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 0.450nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 0.930nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Compound was evaluated for the stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing the 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Compound was evaluated for the stimulation of [35S]GTP-gamma-S, binding in CHO cells expressing the 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 369nMAssay Description:Tested for 5-hydroxytryptamine 1D like receptor-mediated vascular effect in rabbit saphenous vein (RSV)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Tested for 5-hydroxytryptamine 1D like receptor-mediated vascular effect in rabbit saphenous vein (RSV)More data for this Ligand-Target Pair
Affinity DataEC50: 5.10nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist induced [35S]GTP-gamma-S, binding in CHO cells expressing 5-HT 1d receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor beta using rabbit saphenous vein assay.More data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Agonist-induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist-induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist-induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist-induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Agonist-induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 97nMAssay Description:Inhibition of forskolin stimulated adenylate cyclase at 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Effect on forskolin stimulated adenylate cyclase activity at 5-HT1D receptor of guinea pig substantia nigra.More data for this Ligand-Target Pair
Affinity DataEC50: 8.40nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Measurement of agonist induced [35S]GTP-gamma-S, binding in CHO cells stably transfected with 5-hydroxytryptamine 1D receptor.More data for this Ligand-Target Pair
