Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1595
TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332408BDBM332408(US10196353, Example 52 | US11299457, Example 52)
Affinity DataIC50: 15.8nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332406BDBM332406(US10196353, Example 32 | US11299457, Example 32)
Affinity DataIC50: 31.6nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332402BDBM332402(US10196353, Example 17 | US11299457, Example 17)
Affinity DataIC50: 79.4nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332405BDBM332405(US10196353, Example 27 | US11299457, Example 27)
Affinity DataIC50: 79.4nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332052BDBM332052(US10196353, Example 2 | US11299457, Example 2)
Affinity DataIC50: 100nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332404BDBM332404(US10196353, Example 22 | US11299457, Example 22)
Affinity DataIC50: 158nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332401BDBM332401(US10196353, Example 12 | US11299457, Example 12)
Affinity DataIC50: 251nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332403BDBM332403(US10196353, Example 21 | US11299457, Example 21)
Affinity DataIC50: 316nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332400BDBM332400(US10196353, Example 7 | US11299457, Example 7)
Affinity DataIC50: 631nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProgesterone receptor(Human)
Glaxosmithkline

US Patent
LigandChemical structure of BindingDB Monomer ID 332407BDBM332407(US10196353, Example 43 | US11299457, Example 43)
Affinity DataIC50: 631nMAssay Description:Compounds are added to the 384 well black low-volume plates to a final volume of 0.1 μL. DTT and DMSO are added to the chilled assay buffer just...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent