Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50008713
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076389((1S,2S)-2-[(R)-Amino-carboxy-(9-methyl-9H-xanthen-...)
Affinity DataIC50:  34nMAssay Description:Inhibitory activity of the compound against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50049748((2S,4S)-2-Amino-4-(4,4-diphenyl-butyl)-pentanedioi...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity of the compound against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity of the compound against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50052256((S)-3-(amino(carboxy)methyl)bicyclo[1.1.1]pentane-...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50053585((S)-4-(amino(carboxy)methyl)-2-hydroxybenzoic acid...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076392((1S,2S)-2-((S)-1-Amino-1-carboxy-ethyl)-cyclopropa...)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076395((1R,2S,4R)-4-Amino-cyclopentane-1,2,4-tricarboxyli...)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076390((S)-2-Amino-4-carboxy-pentanedioic acid | CHEMBL38...)
Affinity DataIC50:  1.02E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076395((1R,2S,4R)-4-Amino-cyclopentane-1,2,4-tricarboxyli...)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50052256((S)-3-(amino(carboxy)methyl)bicyclo[1.1.1]pentane-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076394(2-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50034503((1R,2R)-3-((S)-Amino-carboxy-methyl)-cyclopropane-...)
Affinity DataIC50:  3.89E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50056272((1S,2S,5R,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dic...)
Affinity DataIC50:  4.58E+5nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076391(7-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076391(7-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory activity of the compound against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed