Affinity DataKi: 0.0100nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-ZM 241385 from Human Adenosine A2a receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 97.6nMAssay Description:Binding affinity against rat adenosine A2A receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Displacement of [3H]-ZM 241385 from Human Adenosine A2a receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 226nMAssay Description:Binding affinity against rat adenosine A1 receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 381nMAssay Description:Displacement of [3H]-ZM 241385 from Human Adenosine A2a receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 594nMAssay Description:Displacement of [3H]-ZM 241385 from Human Adenosine A2a receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against rat adenosine A3 receptor in RBL-2H3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A2B receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-DPCPX from Human Adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair