Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50012876
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM21279(N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123685(4-Bromo-5-(4-chloro-phenyl)-1-(2,4-dichloro-phenyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123690(1-(2,4-Dichloro-phenyl)-5-(4-methoxy-phenyl)-4-met...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123688(4-Bromo-1-(2,4-dichloro-phenyl)-5-(4-methoxy-pheny...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123693(4-Bromo-1-(2-chloro-phenyl)-5-(4-methoxy-phenyl)-1...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123689(1-(2,4-Dichloro-phenyl)-5-(4-methoxy-phenyl)-4-met...)
Affinity DataKi:  7nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123691(5-Benzo[1,3]dioxol-5-yl-1-(2,4-dichloro-phenyl)-4-...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123684(1-(2-Chloro-phenyl)-5-(4-methoxy-phenyl)-4-methyl-...)
Affinity DataKi:  8nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123692(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piper...)
Affinity DataKi:  9nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123683(1-(2-Chloro-phenyl)-4-fluoro-5-(4-methoxy-phenyl)-...)
Affinity DataKi:  18.2nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123687(1-(2-Fluoro-phenyl)-5-(4-methoxy-phenyl)-4-methyl-...)
Affinity DataKi:  37.8nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123694(1-(2,4-Dichloro-phenyl)-5-(4-hydroxy-phenyl)-4-met...)
Affinity DataKi:  104nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123682(1-(2,4-Dichloro-phenyl)-5-(4-methoxy-phenyl)-4-met...)
Affinity DataKi:  380nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50123686(5-(4-Methoxy-phenyl)-1-(2-methoxy-phenyl)-4-methyl...)
Affinity DataKi:  440nMAssay Description:Binding affinity was determined by using a competition assay with [125 I]- AM251 against rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed