Affinity DataKi: 2.70nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.21E+3nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.57E+3nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of 3[H]ATRA binding to retinoid acid receptor gamma expressed in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 259nMAssay Description:Agonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 167nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 143nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 249nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 359nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 6.40nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 3.10nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.80nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.84E+3nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 806nMAssay Description:Inhibition of 3[H]-9-cis-retinoic acid binding to Retinoic acid receptor RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 9.20nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.71E+3nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.40nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Synergistic activation of BRL49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Eli Lilly
Curated by ChEMBL
Eli Lilly
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Antagonist activity against Retinoic acid receptor RXR-alpha expressed in CV-1 cell transcriptional activation assayMore data for this Ligand-Target Pair