Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50013655
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133053(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133054(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133051(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133050(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133054(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  1.03nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133053(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  1.24nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133052(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  1.73nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133055(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133055(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  3.24nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133054(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  3.56nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133053(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133049(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  4.69nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133051(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  5.20nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133053(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  6.57nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50079413(Opioid Peptide [d-Ala(8)]Dynorphin derivative | Ty...)
Affinity DataKi:  8.91nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133056(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  9.54nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133051(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  13.7nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133048(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  26.5nMAssay Description:Binding affinity towards rat Opioid receptor kappa 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]diprenorphine as radiol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133049(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  29.4nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133050(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  32.9nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133055(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  36.5nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133052(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  46.9nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133052(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  47nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133054(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  56.1nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133050(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  72.4nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133056(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  88.3nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50079413(Opioid Peptide [d-Ala(8)]Dynorphin derivative | Ty...)
Affinity DataKi:  123nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133055(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  157nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133051(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  190nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133049(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  206nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133048(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  364nMAssay Description:Binding affinity towards rat Opioid receptor mu 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50079413(Opioid Peptide [d-Ala(8)]Dynorphin derivative | Ty...)
Affinity DataEC50:  515nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133056(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataEC50:  573nMAssay Description:Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133049(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  3.59E+3nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133052(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi:  5.57E+3nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133050(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50079413(Opioid Peptide [d-Ala(8)]Dynorphin derivative | Ty...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133056(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50133048(Opioid Peptide [d-Ala(8)]Dynorphin derivative | CH...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards mouse Opioid receptor delta 1 expressed in CHO cells of chinese hamster ovary was determined using [3H]-DPDGE as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed