Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50037216
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135908(CHEMBL146858 | Cyanonilutamide | 4-(4,4-Dimethyl-2...)
Affinity DataIC50: 6nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135912(5,5-dimethyl-3-[4-nitro-3-(trifluoromethyl)phenyl]...)
Affinity DataIC50: 9nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135914(5-{4-[3-(4-Cyano-3-trifluoromethyl-phenyl)-5,5-dim...)
Affinity DataIC50: 49nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135910(5-(2-{2-[3-(4-Cyano-3-trifluoromethyl-phenyl)-5,5-...)
Affinity DataIC50: 77nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50409765(CHEMBL2112885)
Affinity DataIC50: 90nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50131270(2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]prop...)
Affinity DataIC50: 154nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135911(5-[2-(2-{2-[3-(4-Cyano-3-trifluoromethyl-phenyl)-5...)
Affinity DataIC50: 332nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135915(5-{2-[4-(2-{2-[3-(4-Cyano-3-trifluoromethyl-phenyl...)
Affinity DataIC50: 346nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50135909(5-[2-(4-{4-[3-(4-Cyano-3-trifluoromethyl-phenyl)-5...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Colorado

Curated by ChEMBL
LigandPNGBDBM50056900(2-Carbamoylphenol | 2-Carboxamidophenol | 2-Hydrox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 1.0 nM [3H]mibolerone binding to human androgen receptor of PC3/AR cell lysateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed