Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50042230
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM81471(NSC_5587 | CAS_91-81-6 | Tripelennamine)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataIC50: 158nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422502(CHEMBL158352)
Affinity DataIC50: 251nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422503(CHEMBL157217)
Affinity DataIC50: 398nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422500(CHEMBL157273)
Affinity DataIC50: 398nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50407521(CHEMBL94249)
Affinity DataIC50: 501nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422494(CHEMBL152126)
Affinity DataIC50: 631nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22864(2-[2-(3,3-diphenylpropyl)-1H-imidazol-4-yl]ethan-1...)
Affinity DataIC50: 794nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422495(CHEMBL155188)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50403672(CHEMBL24665)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422496(CHEMBL156071)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422497(CHEMBL152122)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM22865(2-(2-aminoethyl)pyridine | 2-(pyridin-2-yl)ethan-1...)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422504(CHEMBL155314)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM86172(2-(3-Chlorophenyl)histamine)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422501(CHEMBL345185)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422493(CHEMBL359122)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422506(CHEMBL157842)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50407520(CHEMBL90063)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422499(CHEMBL152221)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422498(CHEMBL154566)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50422505(CHEMBL154068)
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed