Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50015549
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50064482(2-demethylthiocolchicine | CHEMBL277239 | N-((S)-2...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157477(CHEMBL142588 | N-((S)-10-Hydroxy-1,2,3-trimethoxy-...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157478(CHEMBL180388 | CHEMBL180503 | Dimethylamino-acetic...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157479(2-Desmethylcolchicin | 2-demethylcolchicine | 2-di...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157478(CHEMBL180388 | CHEMBL180503 | Dimethylamino-acetic...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157480(CHEMBL183373 | CHEMBL183569 | Dimethylamino-acetic...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta-1 chain(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50157480(CHEMBL183373 | CHEMBL183569 | Dimethylamino-acetic...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory concentration against tubulin assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed