Compile Data Set for Download or QSAR
maximum 50k data
Found 55 Enz. Inhib. hit(s) with all data for entry = 50016650
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171546((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  0.720nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171558(2,6-Diamino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  6.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171559((S)-2,3-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  8.20nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against human fibroblast activation protein alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  38nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171557((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-3-m...)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171547((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-but...)
Affinity DataIC50:  49nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  65nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171550((S)-2-Amino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  71nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  95nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171561((S)-2,4-Diamino-4-piperidin-1-yl-butyric acid | CH...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171550((S)-2-Amino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171557((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-3-m...)
Affinity DataIC50:  190nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171549((S)-2-Amino-N-(1-boron-dihydroxide-pentyl)-propion...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171547((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-but...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171558(2,6-Diamino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171558(2,6-Diamino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171547((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-but...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171557((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-3-m...)
Affinity DataIC50:  510nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171546((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  800nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171550((S)-2-Amino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  810nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171560((S)-Pyrrolidine-2-carboxylic acid ((R)-1-boron-dih...)
Affinity DataIC50:  890nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171559((S)-2,3-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171554((S)-2,4-Diamino-N-pentyl-butyramide | CHEMBL194496)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration against human fibroblast activation protein alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171546((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171550((S)-2-Amino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171562((S)-2-Amino-hexanoic acid pentylamide | CHEMBL3728...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171549((S)-2-Amino-N-(1-boron-dihydroxide-pentyl)-propion...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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