Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50017002
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataEC50:  1.10nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  1.5nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  1.70nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataEC50:  2.10nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataEC50:  2.90nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  4.30nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataEC50:  6.90nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  11nMAssay Description:Binding to human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176267((S)-N-(naphthalen-2-ylmethyl)-1-(1H-pyrrolo[2,3-f]...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176266((S)-N-(benzo[d][1,3]dioxol-5-ylmethyl)-1-(1H-pyrro...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  18nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176266((S)-N-(benzo[d][1,3]dioxol-5-ylmethyl)-1-(1H-pyrro...)
Affinity DataEC50:  20nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataEC50:  26nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176264((S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-ami...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176267((S)-N-(naphthalen-2-ylmethyl)-1-(1H-pyrrolo[2,3-f]...)
Affinity DataEC50:  27nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataKi:  31nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176272((S)-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-ami...)
Affinity DataEC50:  32nMAssay Description:Binding to human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176265((S)-1-(5-chloro-1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataEC50:  36nMAssay Description:Binding to human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176270((S)-1-(1H-pyrrolo[3,2-h]isoquinolin-1-yl)propan-2-...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176271((S)-N-(2-chlorobenzyl)-1-(1H-pyrrolo[2,3-f]quinoli...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176266((S)-N-(benzo[d][1,3]dioxol-5-ylmethyl)-1-(1H-pyrro...)
Affinity DataEC50:  42nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176271((S)-N-(2-chlorobenzyl)-1-(1H-pyrrolo[2,3-f]quinoli...)
Affinity DataEC50:  44nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176264((S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-ami...)
Affinity DataEC50:  45nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176267((S)-N-(naphthalen-2-ylmethyl)-1-(1H-pyrrolo[2,3-f]...)
Affinity DataEC50:  52nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataKi:  54nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176270((S)-1-(1H-pyrrolo[3,2-h]isoquinolin-1-yl)propan-2-...)
Affinity DataEC50:  62nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176273((S)-1-(1H-pyrrolo[2,3-f]isoquinolin-1-yl)propan-2-...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176270((S)-1-(1H-pyrrolo[3,2-h]isoquinolin-1-yl)propan-2-...)
Affinity DataEC50:  73nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176271((S)-N-(2-chlorobenzyl)-1-(1H-pyrrolo[2,3-f]quinoli...)
Affinity DataEC50:  74nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataEC50:  75nMAssay Description:Binding to human 5HT2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176274((S)-N-benzyl-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176275((S)-N-(cyclohexylmethyl)-1-(1H-pyrrolo[2,3-f]quino...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176269((S)-N-(1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]5-HT from human 5HT2CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176269((S)-N-(1-(1H-pyrrolo[2,3-f]quinolin-1-yl)propan-2-...)
Affinity DataEC50:  91nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176274((S)-N-benzyl-1-(1H-pyrrolo[2,3-f]quinolin-1-yl)pro...)
Affinity DataEC50:  97nMAssay Description:Binding to human 5HT2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176264((S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-ami...)
Affinity DataEC50:  97nMAssay Description:Binding to human 5HT2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis

Curated by ChEMBL
LigandPNGBDBM50176264((S)-1-(1H-pyrrolo[3,2-h]quinolin-1-yl)propan-2-ami...)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]5-HT from human 5HT2BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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