Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50017761
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186127BDBM50186127(N-[(R)-2-{4-[2-(acetyl-ethyl-amino)-1-cyclohexyl-e...)
Affinity DataKi:  2nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186127BDBM50186127(N-[(R)-2-{4-[2-(acetyl-ethyl-amino)-1-cyclohexyl-e...)
Affinity DataKi:  3nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186127BDBM50186127(N-[(R)-2-{4-[2-(acetyl-ethyl-amino)-1-cyclohexyl-e...)
Affinity DataKi:  3nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186131BDBM50186131((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186121BDBM50186121((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclopentyl-...)
Affinity DataKi:  4nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186128BDBM50186128(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(di...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186125BDBM50186125(N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1-(di...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186128BDBM50186128(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(di...)
Affinity DataKi:  5nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186124BDBM50186124(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(N-...)
Affinity DataKi:  6nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186124BDBM50186124(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(N-...)
Affinity DataKi:  6nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186138BDBM50186138(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(N-...)
Affinity DataKi:  7nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186122BDBM50186122(N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1-mor...)
Affinity DataKi:  10nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186120BDBM50186120(N-((R)-3-(4-chlorophenyl)-1-(4-(1-(cyclobutylamino...)
Affinity DataKi:  12nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186135BDBM50186135((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(3-cyclohexyl-1...)
Affinity DataKi:  13nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186119BDBM50186119((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-cycloheptyl-...)
Affinity DataKi:  13nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186133BDBM50186133(3,4-Dihydro-1H-isoquinoline-2-carboxylic acid ((R)...)
Affinity DataKi:  14nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186126BDBM50186126(N-((R)-3-(4-chlorophenyl)-1-(4-(2,6-dimethylheptan...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186132BDBM50186132(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(2,...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186132BDBM50186132(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(2,...)
Affinity DataKi:  18nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50177561BDBM50177561((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamin...)
Affinity DataKi:  20nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186134BDBM50186134(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-2-(me...)
Affinity DataKi:  26nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186130BDBM50186130(N-((R)-3-(4-chlorophenyl)-1-(4-(dicyclohexylmethyl...)
Affinity DataKi:  35nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186118BDBM50186118(N-((R)-3-(4-chlorophenyl)-1-(4-(1-cyclohexyl-3-met...)
Affinity DataKi:  54nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186136BDBM50186136((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-((diethylami...)
Affinity DataKi:  70nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186129BDBM50186129(2-{4-[(R)-3-(4-chloro-phenyl)-2-(2-2,3-dihydro-1H-...)
Affinity DataKi:  148nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186123BDBM50186123(N-((R)-3-(4-chlorophenyl)-1-(4-(1,3-dicyclohexylpr...)
Affinity DataKi:  326nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50186137BDBM50186137((R)-N-((R)-3-(4-chlorophenyl)-1-(4-(1-(diethylamin...)
Affinity DataKi:  3.43E+3nMAssay Description:Inhibition of [125I]NDP-alpha-MSH binding to human MC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed