Compile Data Set for Download or QSAR
Report error Found 126 Enz. Inhib. hit(s) with all data for entry = 50048856
LigandChemical structure of BindingDB Monomer ID 50228318BDBM50228318(CHEMBL279807)
Affinity DataKi:  0.355nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229080BDBM50229080(CHEMBL349665)
Affinity DataKi:  0.457nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229162BDBM50229162(CHEMBL349747)
Affinity DataKi:  0.603nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229147BDBM50229147(CHEMBL348793)
Affinity DataKi:  0.646nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229143BDBM50229143(CHEMBL162971)
Affinity DataKi:  0.661nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229179BDBM50229179(Delequamine)
Affinity DataKi:  0.661nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229152BDBM50229152(CHEMBL349004)
Affinity DataKi:  0.708nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229155BDBM50229155(CHEMBL164420)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229074BDBM50229074(CHEMBL163570)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229171BDBM50229171(CHEMBL411954)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229178BDBM50229178(CHEMBL161278)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229141BDBM50229141(CHEMBL162965)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229149BDBM50229149(CHEMBL159919)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229170BDBM50229170(CHEMBL348831)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229146BDBM50229146(CHEMBL163290)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229077BDBM50229077(CHEMBL348726)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229079BDBM50229079(CHEMBL352278)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229148BDBM50229148(CHEMBL350388)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229072BDBM50229072(CHEMBL162841)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229134BDBM50229134(CHEMBL262446)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229160BDBM50229160(CHEMBL355140)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229137BDBM50229137(CHEMBL350168)
Affinity DataKi:  2nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229138BDBM50229138(CHEMBL162024)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229081BDBM50229081(CHEMBL162109)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229150BDBM50229150(CHEMBL350393)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229139BDBM50229139(CHEMBL349777)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229161BDBM50229161(CHEMBL443554)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229163BDBM50229163(CHEMBL350144)
Affinity DataKi:  5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229157BDBM50229157(CHEMBL346462)
Affinity DataKi:  5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229144BDBM50229144(CHEMBL161070)
Affinity DataKi:  5nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229168BDBM50229168(CHEMBL350105)
Affinity DataKi:  6.30nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229070BDBM50229070(CHEMBL159802)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229166BDBM50229166(CHEMBL435057)
Affinity DataKi:  6.90nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026636BDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229164BDBM50229164(CHEMBL161531)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229078BDBM50229078(CHEMBL354693)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229151BDBM50229151(CHEMBL30477 | WY-26703)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229069BDBM50229069(CHEMBL350312)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50019848BDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  11nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229145BDBM50229145(CHEMBL162686)
Affinity DataKi:  11nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50013515BDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  13nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229075BDBM50229075(CHEMBL160028)
Affinity DataKi:  14nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229169BDBM50229169(CHEMBL160023)
Affinity DataKi:  17nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229167BDBM50229167(CHEMBL351929)
Affinity DataKi:  17nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229071BDBM50229071(CHEMBL354698)
Affinity DataKi:  28nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229176BDBM50229176(CHEMBL161775)
Affinity DataKi:  29nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229174BDBM50229174(CHEMBL350863)
Affinity DataKi:  38nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229158BDBM50229158(CHEMBL350528)
Affinity DataKi:  43nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229172BDBM50229172(CHEMBL163400)
Affinity DataKi:  56nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50229121BDBM50229121(CHEMBL163802)
Affinity DataKi:  58nMAssay Description:Binding affinity to alpha-2 adrenergic receptor determined by measurement of [3H]yohimbine displacement from rat cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2019
Entry Details Article
PubMed
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