Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50025150
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Imperial College

Curated by ChEMBL
LigandPNGBDBM50260259(R(+)-azido(1-(1-phenylethyl)-1H-imidazol-5-yl)meth...)
Affinity DataEC50:  1.10E+4nMAssay Description:Activity at human GABAA alpha-1-beta-2-gamma-2s receptor expressed in HEK293 cells assessed as effect on GABA-induced current at 3 uM by whole cell p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Imperial College

Curated by ChEMBL
LigandPNGBDBM50125935(CHEMBL681 | R(+)-etomidate | Amidate | (R)-1-(1-ph...)
Affinity DataEC50:  1.10E+4nMAssay Description:Activity at human GABAA alpha-1-beta-2-gamma-2s receptor expressed in HEK293 cells assessed as effect on GABA-induced current at 3 uM by whole cell p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)