Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50020179
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories
Curated by ChEMBL
Tanabe Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair





















