Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50020179
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210977BDBM50210977((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210971BDBM50210971((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210992BDBM50210992((R,E)-3-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazi...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210979BDBM50210979((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210977BDBM50210977((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210992BDBM50210992((R,E)-3-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazi...)
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210976BDBM50210976((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210977BDBM50210977((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210972BDBM50210972((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210972BDBM50210972((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210972BDBM50210972((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210982BDBM50210982((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210983BDBM50210983((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210973BDBM50210973((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 15nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210979BDBM50210979((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 17nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210970BDBM50210970((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210970BDBM50210970((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210979BDBM50210979((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208999BDBM50208999(BX-741 | BX-471 | (R)-1-(5-chloro-2-(2-(4-(4-fluor...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208999BDBM50208999(BX-741 | BX-471 | (R)-1-(5-chloro-2-(2-(4-(4-fluor...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210981BDBM50210981((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human CCR1 expressed in THP1 cells assessed as effect on MIP-1-alpha-induced calcium flux by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210982BDBM50210982((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210977BDBM50210977((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 20nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210982BDBM50210982((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 21nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210979BDBM50210979((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 23nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210971BDBM50210971((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 24nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210983BDBM50210983((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 25nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210983BDBM50210983((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210995BDBM50210995((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 26nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210970BDBM50210970((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 26nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210976BDBM50210976((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 38nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210971BDBM50210971((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 39nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210976BDBM50210976((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 42nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210982BDBM50210982((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 47nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210970BDBM50210970((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 49nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210971BDBM50210971((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 50nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210981BDBM50210981((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 54nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208999BDBM50208999(BX-741 | BX-471 | (R)-1-(5-chloro-2-(2-(4-(4-fluor...)
Affinity DataIC50: 59nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210981BDBM50210981((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 63nMAssay Description:Displacement of [125I]MIP1-alpha from human CCR1 expressed in THP1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210978BDBM50210978((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 64nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210988BDBM50210988((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 72nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210986BDBM50210986((R,E)-3-(2-(3-(4-(4-fluorobenzyl)-2-methylpiperazi...)
Affinity DataIC50: 76nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210991BDBM50210991((R)-3-(2-(2-(4-(4-chlorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 78nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210972BDBM50210972((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 87nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210994BDBM50210994((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 90nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50211000BDBM50211000((R)-3-(2-(2-(4-(3,4-difluorobenzyl)-2-methylpipera...)
Affinity DataIC50: 97nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMacrophage inflammatory protein-1 alpha receptor(Rat)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210976BDBM50210976((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 130nMAssay Description:Binding affinity at rat CCR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210989BDBM50210989((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 140nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210998BDBM50210998((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 1(Human)
Tanabe Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50210999BDBM50210999((R)-3-(2-(2-(4-(4-fluorobenzyl)-2-methylpiperazin-...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity against human CCR1 receptor expressed in THP1 cells assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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