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Found 14 Enz. Inhib. hit(s) with all data for entry = 50020299
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212264(3-(3-(4-ethyl-2,2,7-trimethyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  61.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212268(3-(3-(5-ethyl-4-oxo-2,3,4,5-tetrahydro-1H-cyclopen...)
Affinity DataEC50:  96.6nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212269((E)-3-(5-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.20E+3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212271(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  16.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212276(3-(3-(4-ethyl-2,2,7-trimethyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  173nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212281(3-(5-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212273(3-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  24.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212272(3-(3-(5-ethyl-8-methyl-4-oxo-2,3,4,5-tetrahydro-1H...)
Affinity DataEC50:  1.60E+3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212266(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  2.10nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212275(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212267(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  18.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212274(5-((3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetra...)
Affinity DataEC50:  0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212277((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212283((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  67.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed