Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50020321
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212443BDBM50212443((3aR,4R,9aS,E)-7,8-difluoro-4-(2-(5-(3-fluoropheny...)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212440BDBM50212440((3aR,4R,9aS,E)-4-(2-(5-(3-fluorophenyl)pyridin-2-y...)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212436BDBM50212436((3aR,4R,9aS,E)-7-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 7.60nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212429BDBM50212429((3aR,4R,9aS,E)-4-(2-(5-(3-(trifluoromethyl)phenyl)...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212430BDBM50212430((3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212453BDBM50212453((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212445BDBM50212445((3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)...)
Affinity DataIC50: 12.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212438BDBM50212438((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212441BDBM50212441((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 14.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212437BDBM50212437((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 14.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212439BDBM50212439((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 15.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212435BDBM50212435((3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 20.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212431BDBM50212431((3aR,4R,9aS,E)-6,8-difluoro-4-(2-(5-(3-(trifluorom...)
Affinity DataIC50: 21.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212448BDBM50212448((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212444BDBM50212444((3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50: 31.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212454BDBM50212454((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 46.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212455BDBM50212455((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 63.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212456BDBM50212456((3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212446BDBM50212446((3aR,4R,9aS,E)-5-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50: 85.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212432BDBM50212432((3R,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50: 90nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212451BDBM50212451((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-chlorophenyl)py...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212428BDBM50212428((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50: 138nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212447BDBM50212447((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50: 225nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212450BDBM50212450((3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)...)
Affinity DataIC50: 225nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212457BDBM50212457((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-chlorophenyl)py...)
Affinity DataIC50: 328nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212452BDBM50212452((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50: 330nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212442BDBM50212442((3R,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50: 580nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212449BDBM50212449((3S,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50: 3.14E+3nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212434BDBM50212434((3S,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50: 9.17E+3nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50212433BDBM50212433((3aS,4S,9aR,E)-4-(2-(pyridin-2-yl)vinyl)-3a,4,9,9a...)
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed