Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50020321
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212443((3aR,4R,9aS,E)-7,8-difluoro-4-(2-(5-(3-fluoropheny...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212440((3aR,4R,9aS,E)-4-(2-(5-(3-fluorophenyl)pyridin-2-y...)
Affinity DataIC50:  7.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212436((3aR,4R,9aS,E)-7-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  7.60nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212430((3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212429((3aR,4R,9aS,E)-4-(2-(5-(3-(trifluoromethyl)phenyl)...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212453((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212445((3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)...)
Affinity DataIC50:  12.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212438((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212437((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  14.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212441((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  14.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212439((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  15.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212435((3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  20.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212431((3aR,4R,9aS,E)-6,8-difluoro-4-(2-(5-(3-(trifluorom...)
Affinity DataIC50:  21.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212448((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212444((3aR,4R,9aS,E)-6-fluoro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50:  31.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212454((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  46.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212455((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  63.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212456((3aR,4R,9aS,E)-8-fluoro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50:  65nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212446((3aR,4R,9aS,E)-5-fluoro-4-(2-(5-(3-fluorophenyl)py...)
Affinity DataIC50:  85.5nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212432((3R,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50:  90nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212451((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-chlorophenyl)py...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212428((3aR,4R,9aS,E)-6-chloro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50:  138nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212447((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-(trifluoromethy...)
Affinity DataIC50:  225nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212450((3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vinyl)...)
Affinity DataIC50:  225nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212457((3aR,4R,9aS,E)-8-chloro-4-(2-(5-(3-chlorophenyl)py...)
Affinity DataIC50:  328nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212452((3aR,4R,9aS,E)-4-(2-(5-(3-chlorophenyl)pyridin-2-y...)
Affinity DataIC50:  330nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212442((3R,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50:  580nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212449((3S,3aS,4S,9aR,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50:  3.14E+3nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212434((3S,3aR,4R,9aS,E)-4-(2-(6-methoxyquinolin-2-yl)vin...)
Affinity DataIC50:  9.17E+3nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50212433((3aS,4S,9aR,E)-4-(2-(pyridin-2-yl)vinyl)-3a,4,9,9a...)
Affinity DataIC50:  1.20E+4nMAssay Description:Displacement of [3H]haTRAP from PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed