Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50020446
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213931(tylophorinidine | CHEMBL250854)
Affinity DataIC50: 65nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213932([(R)-(+)-deoxytylophorinidine | CHEMBL250474)
Affinity DataIC50: 68nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213934(tylophorinine | CHEMBL398325)
Affinity DataIC50: 110nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213935((12aS,13R)-2,3,6,7-tetramethoxy-9,10,11,12,12a,13-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213936((S)-2,3,6,7-tetramethoxy-8b,9,10,11,12,12a-hexahyd...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213937((12aS,13S)-2,6,7-trimethoxy-9,10,11,12,12a,13-hexa...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213933((12aS,13S)-2,3,6,7-tetramethoxy-9,10,11,12,12a,13-...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213929(tylophoridicine F | CHEMBL401479)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213930(6,7-Dimethoxy-12a-methyl-9,10,11,12,12a,13-hexahyd...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50213938(tylophoridicine C | CHEMBL249029)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed