Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 2483
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21125(Cis-H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]-OH | (5...)
Affinity DataKi:  0.430nM ΔG°:  -53.5kJ/mole EC50:  0.830nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21129((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  0.550nM ΔG°:  -52.9kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21126((5S,8R,10E,13R)-13-[(2S)-2-amino-3-(4-hydroxypheny...)
Affinity DataKi:  0.570nM ΔG°:  -52.8kJ/mole EC50:  0.880nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21129((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  0.822nM ΔG°:  -51.9kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21126((5S,8R,10E,13R)-13-[(2S)-2-amino-3-(4-hydroxypheny...)
Affinity DataKi:  1.30nM ΔG°:  -50.7kJ/mole EC50:  2.65nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21125(Cis-H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]-OH | (5...)
Affinity DataKi:  1.35nM ΔG°:  -50.6kJ/mole EC50:  2.35nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  1.60nM ΔG°:  -50.2kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21127(single bond H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]...)
Affinity DataKi:  7.90nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Universita Degli Studi

LigandPNGBDBM21128(linear H-Tyr-D-AllylGly-Gly-Phe-D-Allylgly-OH | [2...)
Affinity DataKi:  8.10nM ΔG°:  -46.2kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Universita Degli Studi

LigandPNGBDBM21129((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  44.9nM ΔG°:  -41.9kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21127(single bond H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]...)
Affinity DataKi:  56.9nM ΔG°:  -41.4kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21128(linear H-Tyr-D-AllylGly-Gly-Phe-D-Allylgly-OH | [2...)
Affinity DataKi:  64.5nM ΔG°:  -41.0kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Universita Degli Studi

LigandPNGBDBM21126((5S,8R,10E,13R)-13-[(2S)-2-amino-3-(4-hydroxypheny...)
Affinity DataKi:  74.8nM ΔG°:  -40.7kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Universita Degli Studi

LigandPNGBDBM21125(Cis-H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]-OH | (5...)
Affinity DataKi:  576nM ΔG°:  -35.6kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universita Degli Studi

LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  609nM ΔG°:  -35.5kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Universita Degli Studi

LigandPNGBDBM21128(linear H-Tyr-D-AllylGly-Gly-Phe-D-Allylgly-OH | [2...)
Affinity DataKi:  3.87E+3nM ΔG°:  -30.9kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Universita Degli Studi

LigandPNGBDBM21127(single bond H-Tyr-c[D-AllylGly-Gly-Phe-D-Allylgly]...)
Affinity DataKi:  3.96E+3nM ΔG°:  -30.8kJ/molepH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2008
Entry Details Article
PubMed