Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50020832
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218130BDBM50218130(N-tert-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218148BDBM50218148(N-n-butyl-N'-[2-(2-methylphenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218144BDBM50218144(N-tert-butyl-N'-[2-(2-methoxy-4-methylphenoxy)-5-n...)
Affinity DataIC50: 52nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188619BDBM50188619(BM 573 | CHEMBL210602 | N-tert-butyl-N'-[2-(4-meth...)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218139BDBM50218139(N-tert-butyl-N'-[2-(3-bromophenoxy)-5-nitrobenzene...)
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218132BDBM50218132(N-tert-butyl-N'-[2-(3-chlorophenoxy)-5-nitrobenzen...)
Affinity DataIC50: 73nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218141BDBM50218141(N-tert-butyl-N'-[2-(3-iodophenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 95nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218156BDBM50218156(N-n-pentyl-N'-[2-(4-chloroxyphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218128BDBM50218128(N-tert-butyl-N'-[2-(3-methoxyphenoxy)-5-nitrobenze...)
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218131BDBM50218131(N-tert-butyl-N'-[2-(3-methyl-4-chlorophenoxy)-5-ni...)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218137BDBM50218137(N-n-pentyl-N'-[2-(4-bromophenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218152BDBM50218152(N-tert-butyl-N'-[2-(2-bromophenoxy)-5-nitrobenzene...)
Affinity DataIC50: 151nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218145BDBM50218145(N-tert-butyl-N'-[2-(4-methoxyphenoxy)-5-nitrobenze...)
Affinity DataIC50: 152nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218150BDBM50218150(N-n-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 155nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218127BDBM50218127(N-n-pentyl -N'-[2-(2-methylphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 181nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218153BDBM50218153(N-n-pentyl-N'-[2-(3-chlorophenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 201nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218138BDBM50218138(N-tert-butyl-N'-[2-(2-chlorophenoxy)-5-nitrobenzen...)
Affinity DataIC50: 205nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218158BDBM50218158(N-isopropyl-N'-[2-(3-methylphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 205nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218135BDBM50218135(N-n-pentyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 223nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218126BDBM50218126(N-tert-butyl-N'-[2-(2-methylphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 233nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218136BDBM50218136(N-n-pentyl-N'-[2-(4-iodophenoxy)-5-nitrobenzenesul...)
Affinity DataIC50: 302nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50188619BDBM50188619(BM 573 | CHEMBL210602 | N-tert-butyl-N'-[2-(4-meth...)
Affinity DataIC50: 319nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218149BDBM50218149(N-n-pentyl-N'-[2-(2-chlorophenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 387nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218130BDBM50218130(N-tert-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218129BDBM50218129(N-tert-butyl-N'-[2-(4-chlorophenoxy)-5-nitrobenzen...)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218160BDBM50218160(N-tert-butyl-N'-[2-(4-iodophenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 401nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218151BDBM50218151(N-n-pentyl-N'-[2-(3-bromophenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 413nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218146BDBM50218146(N-n-pentyl-N'-[2-(2-bromophenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 423nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218147BDBM50218147(N-n-pentyl-N'-[2-(4-methoxyphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 446nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218125BDBM50218125(N-n-propyl-N'-[2-(4-methylphenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 448nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218141BDBM50218141(N-tert-butyl-N'-[2-(3-iodophenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 470nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218142BDBM50218142(N-isopropyl-N'-[2-(2-methylphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218140BDBM50218140(N-tert-butyl-N'-[2-(4-bromophenoxy)-5-nitrobenzene...)
Affinity DataIC50: 523nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218144BDBM50218144(N-tert-butyl-N'-[2-(2-methoxy-4-methylphenoxy)-5-n...)
Affinity DataIC50: 528nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218124BDBM50218124(N-n-pentyl-N'-[2-(3-methyl-4-chlorophenoxy)-5-nitr...)
Affinity DataIC50: 565nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218143BDBM50218143(N-tert-butyl-N'-[2-(4-methylphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 579nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218148BDBM50218148(N-n-butyl-N'-[2-(2-methylphenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 673nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218139BDBM50218139(N-tert-butyl-N'-[2-(3-bromophenoxy)-5-nitrobenzene...)
Affinity DataIC50: 683nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218132BDBM50218132(N-tert-butyl-N'-[2-(3-chlorophenoxy)-5-nitrobenzen...)
Affinity DataIC50: 698nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218159BDBM50218159(N-n-pentyl-N'-[2-(4-ethoxyphenoxy)-5-nitrobenzenes...)
Affinity DataIC50: 749nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218157BDBM50218157(N-isopropyl-N'-[2-(4-methylphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 843nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218156BDBM50218156(N-n-pentyl-N'-[2-(4-chloroxyphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 871nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218134BDBM50218134(N-tert-butyl-N'-[2-(4-propoxyphenoxy)-5-nitrobenze...)
Affinity DataIC50: 875nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218154BDBM50218154(N-n-pentyl-N'-[2-(3-iodophenoxy)-5-nitrobenzenesul...)
Affinity DataIC50: 885nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218137BDBM50218137(N-n-pentyl-N'-[2-(4-bromophenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218131BDBM50218131(N-tert-butyl-N'-[2-(3-methyl-4-chlorophenoxy)-5-ni...)
Affinity DataIC50: 1.06E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218133BDBM50218133(N-tert-butyl-N'-[2-(4-ethoxyphenoxy)-5-nitrobenzen...)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform beta expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218127BDBM50218127(N-n-pentyl -N'-[2-(2-methylphenoxy)-5-nitrobenzene...)
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218140BDBM50218140(N-tert-butyl-N'-[2-(4-bromophenoxy)-5-nitrobenzene...)
Affinity DataIC50: 1.66E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
University of LièGe

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218150BDBM50218150(N-n-butyl-N'-[2-(3-methylphenoxy)-5-nitrobenzenesu...)
Affinity DataIC50: 1.91E+3nMAssay Description:Antagonist activity at human thromboxane A2 receptor isoform alpha expressed in HEK293 cells assessed as inhibition of U46619-induced calcium mobiliz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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