Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50021342
TargetSodium-dependent serotonin transporter(Human)
Università

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]paroxetine from SERT receptor in human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 2A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50223509((1R,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]paroxetine from SERT receptor in human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223511((1R,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223509((1R,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223511((1R,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223510((1S,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223508((1S,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50223508((1S,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]paroxetine from SERT receptor in human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223509((1R,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50223510((1S,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]paroxetine from SERT receptor in human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223508((1S,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50223510((1S,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50223511((1R,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]paroxetine from SERT receptor in human platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed