Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50038259
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373848(CHEMBL255779)
Affinity DataIC50:  2.30E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373848(CHEMBL255779)
Affinity DataIC50:  4.90E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373844(CHEMBL272948)
Affinity DataIC50:  5.70E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373845(CHEMBL402939)
Affinity DataIC50:  7.80E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373845(CHEMBL402939)
Affinity DataIC50:  9.20E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373844(CHEMBL272948)
Affinity DataIC50:  9.70E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373847(CHEMBL256605)
Affinity DataIC50:  1.57E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373851(CHEMBL256431)
Affinity DataIC50:  1.59E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373851(CHEMBL256431)
Affinity DataIC50:  1.60E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373846(CHEMBL401537)
Affinity DataIC50:  1.97E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373846(CHEMBL401537)
Affinity DataIC50:  2.91E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373847(CHEMBL256605)
Affinity DataIC50:  3.09E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373850(CHEMBL404331)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373849(CHEMBL255988)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50231890(2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl...)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373850(CHEMBL404331)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373849(CHEMBL255988)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50231890(2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl...)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373843(CHEMBL410400)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373843(CHEMBL410400)
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed