Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50025828
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247204(CHEMBL474125 | N-Cyclopropyl-1-(2,4-dichlorophenyl...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247415(5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichloroph...)
Affinity DataKi:  850nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247428(5-(4-Bromophenyl)-N-cyclopropyl-1-(2,4-dichlorophe...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247429(5-(4-Bromophenyl)-N-cycloheptyl-1-(2,4-dichlorophe...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247205(CHEMBL516381 | N-Cycloheptyl-1-(2,4-dichlorophenyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247430(1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidi...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247430(1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidi...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247416(5-(4-Bromophenyl)-1-(2,4-dichlorophenyl)-N-(4-meth...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247390(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(4-met...)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247415(5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichloroph...)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50247416(5-(4-Bromophenyl)-1-(2,4-dichlorophenyl)-N-(4-meth...)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]WIN55212-2 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed