Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50004446
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50483019(CS-023 | R-115685 | R-1558 | R-1L5685 | Ro-4908463...)
Affinity DataIC50: 5.39E+3nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50483019(CS-023 | R-115685 | R-1558 | R-1L5685 | Ro-4908463...)
Affinity DataIC50: 9.85E+3nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50129062(CHEBI:43968 | ICI-194660 | Meropenem | Merrem | Me...)
Affinity DataIC50: 1.38E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50213266(CHEBI:471744 | Imipenem | MK-0787)
Affinity DataIC50: 2.53E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50129062(CHEBI:43968 | ICI-194660 | Meropenem | Merrem | Me...)
Affinity DataIC50: 3.39E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50213266(CHEBI:471744 | Imipenem | MK-0787)
Affinity DataIC50: 5.67E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed