Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 5684
TargetSerine/threonine-protein kinase D1(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 182nMpH: 7.5 T: 2°CAssay Description:The radiometric kinase assay using PKD kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D3(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 227nMpH: 7.5 T: 2°CAssay Description:The radiometric kinase assay using PKD kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D2(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 280nMpH: 7.5 T: 2°CAssay Description:The radiometric kinase assay using PKD kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 500nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
University of Pittsburgh

LigandPNGBDBM92601(CID 797718)
Affinity DataIC50: 2.13E+3nMpH: 7.5 T: 2°CAssay Description:The radiometric kinase assay using PKD kinase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
University of Pittsburgh

LigandPNGBDBM92601(CID 797718)
Affinity DataIC50: 7.00E+3nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
University of Pittsburgh

LigandPNGBDBM92601(CID 797718)
Affinity DataIC50: 8.40E+3nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 1.53E+4nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 2.03E+4nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of Pittsburgh

LigandPNGBDBM92601(CID 797718)
Affinity DataIC50: 2.19E+4nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
University of Pittsburgh

LigandPNGBDBM32334(7-hydroxy-2,3,4,5-tetrahydro-[1]benzofuro[2,3-c]az...)
Affinity DataIC50: 5.00E+4nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
University of Pittsburgh

LigandPNGBDBM92601(CID 797718)
Affinity DataIC50: 5.00E+4nMAssay Description:An IMAP-based PKD HTS FR assay was used for primary HTS of the PMLSC library to identify hit compounds and subsequent secondary hit confirmation stud...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed