Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50028006
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256003BDBM50256003(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 14nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256004BDBM50256004(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 29nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256043BDBM50256043(CHEMBL480350 | Hymenialdisine, 10 | (Z)-3-bromohym...)
Affinity DataIC50: 100nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256000BDBM50256000(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 140nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256025BDBM50256025(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256047BDBM50256047(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256028BDBM50256028(4-[2-Amino-4-oxo-4H-thiazol-(5)-ylidene]-4,6,7,9-t...)
Affinity DataIC50: 180nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256029BDBM50256029(4-[2-Amino-4-oxo-4H-thiazol-(5)-ylidene]-1-bromo-4...)
Affinity DataIC50: 190nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256027BDBM50256027(10-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene...)
Affinity DataIC50: 230nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256008BDBM50256008({5-[1-Bromo-8-oxo-6,7,8,9-tetrahydro-5H-3-thia-7,9...)
Affinity DataIC50: 260nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256030BDBM50256030(1-Bromo-4-[2-(2-hydroxy-ethylamino)-5-oxo-3,5-dihy...)
Affinity DataIC50: 280nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256048BDBM50256048(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 300nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16591BDBM16591(B722657K110 | Hymenialdisine, 8 | CHEMBL255465 | (...)
Affinity DataIC50: 330nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256002BDBM50256002(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 460nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025098BDBM50025098(CHEMBL332551)
Affinity DataIC50: 470nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256001BDBM50256001(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 890nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256026BDBM50256026(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256009BDBM50256009(4-[2-(2-Hydroxy-ethylamino)-5-oxo-3,5-dihydro-imid...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7491BDBM7491(4-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256007BDBM50256007(10-[2-Amino-4-oxo-4H-thiazol-(5)-ylidene]-7,8,9,10...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256006BDBM50256006(4-[2-Amino-4-oxo-4H-thiazol-(5)-ylidene]-1-phenyl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256046BDBM50256046(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Institut De Recherche Servier

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256045BDBM50256045(4-[2-Amino-5-oxo-3,5-dihydro-imidazol-(4)-ylidene]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed