Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50028397
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278254(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 1.35nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278255(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 1.46nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278201(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 1.47nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278136(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 1.66nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278311(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-N-phenyl-...)
Affinity DataIC50: 1.94nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278310(5-(4-bromophenyl)-3-(5-(1-(4-chlorophenyl)cyclopro...)
Affinity DataIC50: 1.96nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278073(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 3.27nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278202(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 3.51nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278820(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 5.72nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278075(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 7.25nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278821(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 9.31nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278204(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 11.5nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278819(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 12.7nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278203(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 13.4nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278076(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 17.2nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278074(N-butyl-3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4...)
Affinity DataIC50: 17.8nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278818(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 18.3nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278747(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 23.8nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278252(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 62.1nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278253((3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chloro...)
Affinity DataIC50: 93.4nMAssay Description:Displacement of [3H]CP-55940 from cannabinoid CB1 receptor in Sprague-Dawley rat cerebellar membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278255(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 374nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278254(5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-oxadiazol-...)
Affinity DataIC50: 386nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278311(5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-N-phenyl-...)
Affinity DataIC50: 488nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278201(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 636nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278136(3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-5-(4-chlorop...)
Affinity DataIC50: 738nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 1.76E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Green Cross

Curated by ChEMBL
LigandPNGBDBM50278310(5-(4-bromophenyl)-3-(5-(1-(4-chlorophenyl)cyclopro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]WIN-55212-2 from human recombinant cannabinoid CB2 receptor expressed in CHOK1 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed