Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 50030281
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293634(CHEMBL569374 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293636(CHEMBL561293 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293623(CHEMBL551841 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293637(CHEMBL551488 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293618(CHEMBL563684 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293613(CHEMBL554742 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293628(CHEMBL561228 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293608(CHEMBL561355 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293639(CHEMBL551693 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293638(CHEMBL560629 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293633(CHEMBL560230 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293631(4-bromo-N-(3-bromo-4-(2-(2-methylpyrrolidin-1-yl)e...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293631(4-bromo-N-(3-bromo-4-(2-(2-methylpyrrolidin-1-yl)e...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293635(CHEMBL571006 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293640(CHEMBL563558 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293622(CHEMBL559766 | N-(3-bromo-4-(2-(dimethylamino)etho...)
Affinity DataKi:  670nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50253285(4-Bromo-N-(3-bromo-4-(3-(dimethylamino)propoxy)phe...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293632(4-bromo-N-(3-bromo-4-(2-(3-fluoropyrrolidin-1-yl)e...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293632(4-bromo-N-(3-bromo-4-(2-(3-fluoropyrrolidin-1-yl)e...)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293625(CHEMBL559963 | N-(3-bromo-4-((1-methylpiperidin-3-...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293610(CHEMBL554516 | N-(3-bromo-4-((1-methylpiperidin-3-...)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293611(CHEMBL561234 | N-(3-bromo-4-(3-(dimethylamino)prop...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293615(CHEMBL564035 | N-(3-bromo-4-((1-methylpiperidin-3-...)
Affinity DataKi:  1.52E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293612(CHEMBL561433 | N-(3-bromo-4-(2-(dimethylamino)etho...)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293621(CHEMBL551840 | N-(3-bromo-4-(3-(dimethylamino)prop...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293607(CHEMBL570774 | N-(3-bromo-4-(2-(dimethylamino)etho...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293620(CHEMBL562235 | N-(3-bromo-4-((1-methylpiperidin-3-...)
Affinity DataKi:  1.65E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293616(CHEMBL561837 | N-(3-bromo-4-(3-(dimethylamino)prop...)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293630(CHEMBL559842 | N-(3-bromo-4-((1-methylpiperidin-3-...)
Affinity DataKi:  2.11E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293617(CHEMBL550141 | N-(3-bromo-4-(2-(dimethylamino)etho...)
Affinity DataKi:  2.13E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293626(CHEMBL554108 | N-(3-bromo-4-(3-(dimethylamino)prop...)
Affinity DataKi:  2.29E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293627(CHEMBL562297 | N-(3-bromo-4-(2-(dimethylamino)etho...)
Affinity DataKi:  2.72E+3nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293609(CHEMBL549332 | N-(3-bromo-4-(2-morpholinoethoxy)ph...)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293624(CHEMBL549544 | N-(3-bromo-4-(2-morpholinoethoxy)ph...)
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293619(CHEMBL561029 | N-(3-bromo-4-(2-morpholinoethoxy)ph...)
Affinity DataKi:  1.76E+4nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293614(CHEMBL563666 | N-(3-bromo-4-(2-morpholinoethoxy)ph...)
Affinity DataKi:  2.64E+4nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293629(CHEMBL559448 | N-(3-bromo-4-(2-morpholinoethoxy)ph...)
Affinity DataKi:  3.25E+4nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293636(CHEMBL561293 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293634(CHEMBL569374 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293623(CHEMBL551841 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293637(CHEMBL551488 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  260nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293618(CHEMBL563684 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293613(CHEMBL554742 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  380nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293628(CHEMBL561228 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  390nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293608(CHEMBL561355 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  430nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293639(CHEMBL551693 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  450nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293638(CHEMBL560629 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  550nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293633(CHEMBL560230 | N-(3-bromo-4-(2-(pyrrolidin-1-yl)et...)
Affinity DataIC50:  560nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293631(4-bromo-N-(3-bromo-4-(2-(2-methylpyrrolidin-1-yl)e...)
Affinity DataIC50:  710nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50293631(4-bromo-N-(3-bromo-4-(2-(2-methylpyrrolidin-1-yl)e...)
Affinity DataIC50:  750nMAssay Description:Displacement of [3H]SMT from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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