Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50028786
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21278BDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268759BDBM50268759(N-butyl-2-chloro-N-(2-(4-(4-chlorophenyl)pyrrolo[1...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268683BDBM50268683(N-butyl-2-chloro-N-(2-(4-(4-methoxyphenyl)pyrrolo[...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268633BDBM50268633(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268634BDBM50268634(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268514BDBM50268514(N-butyl-2-chloro-N-(2-(4-(4-methoxyphenyl)pyrrolo[...)
Affinity DataKi:  137nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268758BDBM50268758(N-butyl-2-chloro-N-(2-(4-(4-fluorophenyl)pyrrolo[1...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268632BDBM50268632(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268454BDBM50268454(2-chloro-N-isopropyl-N-(2-(4-(4-methoxyphenyl)pyrr...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268569BDBM50268569(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  236nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268721BDBM50268721(N-butyl-2-chloro-N-(2-oxo-2-(4-phenylpyrrolo[1,2-a...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268568BDBM50268568(N-butyl-2-fluoro-N-(2-(4-(4-methoxyphenyl)pyrrolo[...)
Affinity DataKi:  349nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268682BDBM50268682(N-butyl-2-methoxy-N-(2-(4-(4-methoxyphenyl)pyrrolo...)
Affinity DataKi:  461nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268567BDBM50268567(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268681BDBM50268681(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  539nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268570BDBM50268570(N-butyl-N-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]qui...)
Affinity DataKi:  602nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50268513BDBM50268513(N-butyl-3,5-dichloro-N-(2-(4-(4-methoxyphenyl)pyrr...)
Affinity DataKi:  831nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed