Compile Data Set for Download or QSAR
Report error Found 208 Enz. Inhib. hit(s) with all data for entry = 50030354
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294961BDBM50294961(1-(2-Chloro-4-(hexylsulfonyl)phenyl)-3-(4-(ethylsu...)
Affinity DataIC50: 400nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294962BDBM50294962(3-(4-Acetylpiperazin-1-yl)-1-(2-chloro-4-(hexylsul...)
Affinity DataIC50: 500nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294963BDBM50294963(1-(2,5-Dichloro-4-(hexyloxy)phenyl)-3-(dimethylami...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to TRalpha receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294963BDBM50294963(1-(2,5-Dichloro-4-(hexyloxy)phenyl)-3-(dimethylami...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294964BDBM50294964(3-(4-Acetylpiperazin-1-yl)-1-(2,3-dichloro-4-(hexy...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294967BDBM50294967(4-(3-(2,5-Dichloro-4-(hexylthio)phenyl)-3-oxopropy...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294968BDBM50294968(1-(2-Chloro-4-(hexylsulfonyl)phenyl)-3-morpholinop...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294965BDBM50294965(3-(4-acetylpiperazin-1-yl)-1-(2,6-dichloro-4-(hexy...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294966BDBM50294966(3-(4-Acetylpiperazin-1-yl)-1-(2-chloro-4-(hexylthi...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294969BDBM50294969(4-(3-(2,5-Dichloro-4-(hexylsulfonyl)phenyl)-3-oxop...)
Affinity DataIC50: 600nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294970BDBM50294970(1-(2,6-dichloro-4-(hexyloxy)phenyl)-3-(dimethylami...)
Affinity DataIC50: 690nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294975BDBM50294975(1-(2,3-Dichloro-4-(hexylsulfonyl)phenyl)-3-morphol...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294976BDBM50294976(3-(4-acetylpiperazin-1-yl)-1-(2,6-dichloro-4-(hexy...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294973BDBM50294973(1-(2,5-Dichloro-4-(hexylthio)phenyl)-3-(4-(ethylsu...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294974BDBM50294974(4-(3-(2-Chloro-4-(hexylsulfonyl)phenyl)-3-oxopropy...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294895BDBM50294895(3-(Dimethylamino)-1-(4-(hexyloxy)-2,6-dimethylphen...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294971BDBM50294971(1-(2,3-Dichloro-4-(hexyloxy)phenyl)-3-morpholinopr...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294972BDBM50294972(1-(2,3-Dichloro-4-(hexylthio)phenyl)-3-(4-(ethylsu...)
Affinity DataIC50: 700nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294979BDBM50294979(1-(2,6-dichloro-4-(hexyloxy)phenyl)-3-(4-(ethylsul...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294980BDBM50294980(1-(2-Chloro-4-(hexylthio)phenyl)-3-morpholinopropa...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294977BDBM50294977(3-(4-Acetylpiperazin-1-yl)-1-(2,5-dichloro-4-(hexy...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294978BDBM50294978(1-(2,6-dichloro-4-(hexyloxy)phenyl)-3-morpholinopr...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294983BDBM50294983(4-(3-(2,3-Dichloro-4-(hexylsulfonyl)phenyl)-3-oxop...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294984BDBM50294984(3-(4-Acetylpiperazin-1-yl)-1-(2,5-dichloro-4-(hexy...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294981BDBM50294981(4-(3-(2,3-Dichloro-4-(hexylthio)phenyl)-3-oxopropy...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294982BDBM50294982(3-(4-Acetylpiperazin-1-yl)-1-(2,5-dichloro-4-(hexy...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294987BDBM50294987(1-(2,6-dichloro-4-(hexylsulfonyl)phenyl)-3-(4-(eth...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294985BDBM50294985(1-(2,5-Dichloro-4-(hexylsulfonyl)phenyl)-3-(4-(eth...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294986BDBM50294986(1-(2,6-dichloro-4-(hexylsulfonyl)phenyl)-3-morphol...)
Affinity DataIC50: 800nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294996BDBM50294996(1-(2,3-dichloro-4-(hexyloxy)phenyl)-3-(dimethylami...)
Affinity DataIC50: 810nMAssay Description:Inhibition of SRC2 binding to TRalpha receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294991BDBM50294991(1-(2,5-Dichloro-4-(hexylsulfonyl)phenyl)-3-morphol...)
Affinity DataIC50: 900nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294992BDBM50294992(1-(4-(Hexylsulfonyl)-2,6-dimethylphenyl)-3-morphol...)
Affinity DataIC50: 900nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294989BDBM50294989(3-(4-Acetylpiperazin-1-yl)-1-(4-(hexylthio)-2,6-di...)
Affinity DataIC50: 900nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294990BDBM50294990(1-(2,3-Dichloro-4-(hexylsulfonyl)phenyl)-3-(4-(eth...)
Affinity DataIC50: 900nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294988BDBM50294988(3-(4-Acetylpiperazin-1-yl)-1-(2,3-dichloro-4-(hexy...)
Affinity DataIC50: 900nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294995BDBM50294995(4-(3-(2,6-dichloro-4-(hexylsulfonyl)phenyl)-3-oxop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294993BDBM50294993(1-(2,5-Dichloro-4-(hexylthio)phenyl)-3-morpholinop...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294994BDBM50294994(3-(4-Acetylpiperazin-1-yl)-1-(2,3-dichloro-4-(hexy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294996BDBM50294996(1-(2,3-dichloro-4-(hexyloxy)phenyl)-3-(dimethylami...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294887BDBM50294887(1-(2-Bromo-4-(hexyloxy)phenyl)-3-(dimethylamino)pr...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to TRalpha receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294999BDBM50294999(1-(2,6-Dichloro-4-(hexylsulfonyl)phenyl)-3-(dimeth...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295000BDBM50295000(3-(Dimethylamino)-1-(4-(hexylsulfonyl)-2,6-dimethy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294997BDBM50294997(1-(2,6-Dichloro-4-(hexylthio)phenyl)-3-morpholinop...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294998BDBM50294998(3-(4-Acetylpiperazin-1-yl)-1-(2,6-dichloro-4-(hexy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295005BDBM50295005(1-(2,3-Dichloro-4-(hexylsulfonyl)phenyl)-3-(2-meth...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294919BDBM50294919(3-(Dimethylamino)-1-(4-(hexyloxy)-3-iodophenyl)pro...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to TRalpha receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50294931BDBM50294931(3-(4-Acetylpiperazin-1-yl)-1-(4-(hexylsulfonyl)-2,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295003BDBM50295003(1-(2,3-Dichloro-4-(hexyloxy)phenyl)-3-(4-(ethylsul...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295004BDBM50295004(1-(2,5-Dichloro-4-(hexylthio)phenyl)-3-(dimethylam...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
St. Jude Children'S Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295001BDBM50295001(3-(4-Acetylpiperazin-1-yl)-1-(2-chloro-4-(hexyloxy...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SRC2 binding to human TRbeta receptor ligand binding domain expressed in Escherichia coli BL21 (DE3) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
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