Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50030430
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296045(N-(1-(6-oxo-1,6-dihydropyridin-3-yl)pentyl)-2-(1-(...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296041(N-((4-fluorophenyl)(6-methoxypyridin-3-yl)methyl)-...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296044(N-((4-fluorophenyl)(6-oxo-1,6-dihydropyridin-3-yl)...)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296019(N-(4-fluorobenzyl)-N-(3-hydroxypropyl)-2-(1-((1-(4...)
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296042(N-(1-(6-methoxypyridin-3-yl)pentyl)-2-(1-((1-(4-(t...)
Affinity DataIC50: 5nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296043(N-((5-chloro-6-oxo-1,6-dihydropyridin-3-yl)(4-fluo...)
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296047(N-(2,4-dichlorobenzyl)-4-((1-(4-(trifluoromethyl)p...)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296017(N-(bis(4-fluorophenyl)methyl)-2-(1-((1-(5-(trifluo...)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296038(N-((4-chlorophenyl)(pyridin-4-yl)methyl)-2-(1-((1-...)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296035(N-((1H-imidazol-5-yl)(phenyl)methyl)-2-(1-((1-(4-(...)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296017(N-(bis(4-fluorophenyl)methyl)-2-(1-((1-(5-(trifluo...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296045(N-(1-(6-oxo-1,6-dihydropyridin-3-yl)pentyl)-2-(1-(...)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296043(N-((5-chloro-6-oxo-1,6-dihydropyridin-3-yl)(4-fluo...)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296040(3-((4-fluorophenyl)(2-(1-((1-(4-(trifluoromethyl)p...)
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296025(N-(4-chloro-2-hydroxybenzyl)-1-((1-(4-(trifluorome...)
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296044(N-((4-fluorophenyl)(6-oxo-1,6-dihydropyridin-3-yl)...)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human MCHR1 expressed in HEK293 cells assessed as [35S]GTPgammaS accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296039(N-((4-fluorophenyl)(pyridin-3-yl)methyl)-2-(1-((1-...)
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50245454(2-(3-chlorophenoxy)-N-(1-((1-(4-(trifluoromethyl)p...)
Affinity DataIC50: 29nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296024(N-(2-chloro-4-hydroxybenzyl)-1-((1-(4-(trifluorome...)
Affinity DataIC50: 30nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296030(N,N-diethyl-1-(2-(1-((1-(4-(trifluoromethyl)phenyl...)
Affinity DataIC50: 37nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296048(1-benzhydryl-3-(1-((1-(4-(trifluoromethyl)phenyl)-...)
Affinity DataIC50: 39nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296023(N-((1-hydroxycyclohexyl)methyl)-1-((1-(4-(trifluor...)
Affinity DataIC50: 40nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296037(N-(phenyl(pyridin-2-yl)methyl)-2-(1-((1-(4-(triflu...)
Affinity DataIC50: 41nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296016(N-(bis(4-fluorophenyl)methyl)-2-(4-((1-(5-(trifluo...)
Affinity DataIC50: 55nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296036(N-(2-(2-methyl-1H-imidazol-1-yl)-1-phenylethyl)-2-...)
Affinity DataIC50: 65nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296032(1-(2-(pyrrolidine-1-carbonyl)piperidin-1-yl)-2-(1-...)
Affinity DataIC50: 66nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296046(N-(1-(6-oxo-1,6-dihydropyridin-3-yl)ethyl)-2-(1-((...)
Affinity DataIC50: 67nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296031(1-(3-(pyrrolidine-1-carbonyl)piperidin-1-yl)-2-(1-...)
Affinity DataIC50: 71nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296029(N-methyl-N-(3-oxo-3-(pyrrolidin-1-yl)propyl)-2-(1-...)
Affinity DataIC50: 142nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296026(N-(2,4-dichloro-6-hydroxybenzyl)-1-((1-(4-(trifluo...)
Affinity DataIC50: 144nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296020(2-(1-((5-(4-chlorophenyl)furan-2-yl)methyl)piperid...)
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296033(1-(2-(pyrrolidine-1-carbonyl)morpholino)-2-(1-((1-...)
Affinity DataIC50: 173nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296028(N-((1-methyl-1H-pyrrol-2-yl)methyl)-2-(1-((1-(4-(t...)
Affinity DataIC50: 313nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296027(N-(2-(pyridin-2-yl)ethyl)-1-((1-(4-(trifluoromethy...)
Affinity DataIC50: 339nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296034(1-(4-(pyrrolidine-1-carbonyl)piperazin-1-yl)-2-(1-...)
Affinity DataIC50: 417nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296018(N-(2,4-dichlorobenzyl)-1-((1-(5-(trifluoromethyl)p...)
Affinity DataIC50: 444nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50245454(2-(3-chlorophenoxy)-N-(1-((1-(4-(trifluoromethyl)p...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296022(2-(1-((5-(4-chlorophenyl)furan-2-yl)methyl)piperid...)
Affinity DataIC50: 597nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296019(N-(4-fluorobenzyl)-N-(3-hydroxypropyl)-2-(1-((1-(4...)
Affinity DataIC50: 630nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296017(N-(bis(4-fluorophenyl)methyl)-2-(1-((1-(5-(trifluo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296016(N-(bis(4-fluorophenyl)methyl)-2-(4-((1-(5-(trifluo...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296021(2-(1-((5-(4-chlorophenyl)furan-2-yl)methyl)piperid...)
Affinity DataIC50: 815nMAssay Description:Displacement of [125I]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296042(N-(1-(6-methoxypyridin-3-yl)pentyl)-2-(1-((1-(4-(t...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296021(2-(1-((5-(4-chlorophenyl)furan-2-yl)methyl)piperid...)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296020(2-(1-((5-(4-chlorophenyl)furan-2-yl)methyl)piperid...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296025(N-(4-chloro-2-hydroxybenzyl)-1-((1-(4-(trifluorome...)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296024(N-(2-chloro-4-hydroxybenzyl)-1-((1-(4-(trifluorome...)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296047(N-(2,4-dichlorobenzyl)-4-((1-(4-(trifluoromethyl)p...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG activation expressed in CHO cells by rubidium efflux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296038(N-((4-chlorophenyl)(pyridin-4-yl)methyl)-2-(1-((1-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca R & D M£Lndal

Curated by ChEMBL
LigandPNGBDBM50296041(N-((4-fluorophenyl)(6-methoxypyridin-3-yl)methyl)-...)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
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