Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50004390
Target3-phosphoinositide-dependent protein kinase 1(Human)
Universit£Tsklinikum Frankfurt

Curated by ChEMBL
LigandPNGBDBM50296954((Z)-5-(4-bromo-2-fluorophenyl)-3-phenylpent-2-enoi...)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to human PDPK1 Y288G/Q292A mutant expressed in insect cell system assessed as substrate phosphorylation by isothermal titration calo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target3-phosphoinositide-dependent protein kinase 1(Human)
Universit£Tsklinikum Frankfurt

Curated by ChEMBL
LigandPNGBDBM50296949(PS48 | (2Z)-5-(4-chlorophenyl)-3-phenylpent-2-enoi...)
Affinity DataKd:  1.03E+4nMAssay Description:Binding affinity to human PDPK1 Y288G/Q292A mutant expressed in insect cell system assessed as substrate phosphorylation by isothermal titration calo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)