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Found 17 Enz. Inhib. hit(s) with all data for entry = 50035890
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010707(8-Chloro-3-methyl-5-m-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Mus musculus (Mouse))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010717(8-Chloro-3-methyl-5-o-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010716(8-Chloro-3-methyl-5-p-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004823((6aS,13bR)-11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004822((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010709(5-Benzofuran-7-yl-8-chloro-3-methyl-2,3,4,5-tetrah...)
Affinity DataKi:  6nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004820(3-Chloro-7-methyl-5,6,7,7a,8,12b-hexahydro-7-aza-d...)
Affinity DataKi:  7nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010708(6-Phenyl-2,6,7,8,9,9a-hexahydro-1H-8-aza-benzo[cd]...)
Affinity DataKi:  24nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  192nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010715((6aS,13bS)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahy...)
Affinity DataKi:  513nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010711((6aR,13bS )11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  531nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010712((6aR,13bR)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahy...)
Affinity DataKi:  898nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010710(6-Phenyl-2,6,7,8,9,9a-hexahydro-1H-8-aza-benzo[cd]...)
Affinity DataKi:  1.22E+3nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 5(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010714(1-p-Tolyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,...)
Affinity DataEC50:  210nMAssay Description:Effective concentration required to stimulate Adenylate cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 5(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004822((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)
Affinity DataEC50:  80nMAssay Description:Effective concentration required to stimulate Adenylate cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed