Affinity DataKi: 0.300nMAssay Description:Binding affinity to human NK3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]osanetant from human recombinant NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Displacement of [3H]osanetant from guinea pig recombinant NK3 receptor A1142.58T expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 35.5nMAssay Description:Displacement of [3H]SR48968 from human recombinant NK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 70.9nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 109nMAssay Description:Displacement of [3H]SR48968 from human recombinant NK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 515nMAssay Description:Displacement of [3H]SR48968 from human recombinant NK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 953nMAssay Description:Displacement of [3H]SR48968 from human recombinant NK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity to human NK2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR48968 from human recombinant NK2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at guinea pig NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphateMore data for this Ligand-Target Pair
Affinity DataKd: 0.0800nMAssay Description:Apparent binding affinity to guinea pig NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.150nMAssay Description:Equilibrium binding affinity to guinea pig NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at human NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphateMore data for this Ligand-Target Pair
Affinity DataKd: 0.200nMAssay Description:Equilibrium binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.220nMAssay Description:Apparent binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair