Compile Data Set for Download or QSAR
maximum 50k data
Found 85 Enz. Inhib. hit(s) with all data for entry = 50031047
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305980((S)-2-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)-3-...)
Affinity DataIC50:  500nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305909((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-(methylth...)
Affinity DataIC50:  500nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305923((S)-2-(4-chlorophenyl)-4-methyl-N-(thiazol-2-yl)pe...)
Affinity DataIC50:  600nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305904((S)-2-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)-3,...)
Affinity DataIC50:  700nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305981((S)-2-(4-chlorophenyl)-N-(5-chlorothiazol-2-yl)-3-...)
Affinity DataIC50:  700nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305906((S)-N-(5-bromothiazol-2-yl)-2-(4-chlorophenyl)-3,3...)
Affinity DataIC50:  700nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305974((S)-2-(4-chlorophenyl)-3-methyl-N-(thiazol-2-yl)bu...)
Affinity DataIC50:  700nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305911((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-phenylthi...)
Affinity DataIC50:  700nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305973(2-(4-chlorophenyl)-3-methyl-N-(thiazol-2-yl)butana...)
Affinity DataIC50:  800nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305979((S)-2-(4-chlorophenyl)-3-methyl-N-(5-methylthiazol...)
Affinity DataIC50:  800nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305905((S)-2-(4-chlorophenyl)-N-(5-chlorothiazol-2-yl)-3,...)
Affinity DataIC50:  1.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305950((S)-2-(4-chlorophenyl)-N-(6-fluoropyridin-2-yl)-3-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305926((S)-2-(4-chlorophenyl)-N-(thiazol-2-yl)pent-4-enam...)
Affinity DataIC50:  1.10E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305933((S)-2-cyclopropyl-N-(5-fluorothiazol-2-yl)-2-(4-(t...)
Affinity DataIC50:  1.10E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305922((S)-2-(4-chlorophenyl)-2-cyclopropyl-N-(5-fluoroth...)
Affinity DataIC50:  1.20E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305917((S)-2-(4-chlorophenyl)-N-(5-(1,1,1,3,3,3-hexafluor...)
Affinity DataIC50:  1.20E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305951((S)-2-(4-chlorophenyl)-N-(5-fluoropyridin-2-yl)-3-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305949((S)-2-(4-chlorophenyl)-3-methyl-N-(pyridin-2-yl)bu...)
Affinity DataIC50:  1.40E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305969((S)-2-(4-chlorophenyl)-3-methyl-N-(4-methylthiazol...)
Affinity DataIC50:  1.40E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305908((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-(trifluor...)
Affinity DataIC50:  1.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305907((S)-2-(4-chlorophenyl)-N-(5-cyanothiazol-2-yl)-3,3...)
Affinity DataIC50:  1.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305982((S)-2-(4-chlorophenyl)-3-methyl-N-(5-(trifluoromet...)
Affinity DataIC50:  1.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305930(1-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)cyclobu...)
Affinity DataIC50:  1.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305914((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-morpholin...)
Affinity DataIC50:  1.60E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305913((S)-2-(4-chlorophenyl)-N-(5-(dimethylamino)thiazol...)
Affinity DataIC50:  1.60E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305978((S)-2-(4-chlorophenyl)-N-(4,5-dimethylthiazol-2-yl...)
Affinity DataIC50:  1.80E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305957((S)-2-(4-chlorophenyl)-3-methyl-N-(5-(trifluoromet...)
Affinity DataIC50:  1.90E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305901((S)-2-(4-chlorophenyl)-N-(5-cyanothiazol-2-yl)-3-m...)
Affinity DataIC50:  2.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305902((S)-methyl 2-(2-(4-chlorophenyl)-3-methylbutanamid...)
Affinity DataIC50:  2.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305958((S)-2-(4-chlorophenyl)-3-methyl-N-(1,2,4-thiadiazo...)
Affinity DataIC50:  2.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305964((S)-2-(4-chlorophenyl)-N-(4,5-dihydrothiazol-2-yl)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305954((S)-2-(4-chlorophenyl)-3-methyl-N-(pyridazin-3-yl)...)
Affinity DataIC50:  2.30E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305916((S)-2-(4-Chloro-phenyl)-N-[5-(1,1-dioxo-1lambda*6*...)
Affinity DataIC50:  2.40E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305966(CHEMBL609852 | rac-N-(benzo[d]thiazol-2-yl)-2-(4-c...)
Affinity DataIC50:  3.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305910((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-(methylsu...)
Affinity DataIC50:  3.40E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305915((S)-2-(4-chlorophenyl)-3,3-dimethyl-N-(5-(4-methyl...)
Affinity DataIC50:  3.80E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305967((S)-N-(5-chlorobenzo[d]oxazol-2-yl)-2-(4-chlorophe...)
Affinity DataIC50:  4.30E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305931(1-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)cyclope...)
Affinity DataIC50:  5.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305920((S)-2-(4-chlorophenyl)-N-(thiazol-2-yl)butanamide ...)
Affinity DataIC50:  5.00E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305968(CHEMBL610060 | rac-N-(1H-benzo[d]imidazol-2-yl)-2-...)
Affinity DataIC50:  5.20E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305921((S)-2-(4-chlorophenyl)-N-(thiazol-2-yl)pentanamide...)
Affinity DataIC50:  5.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305953(CHEMBL611632 | rac-2-(4-chlorophenyl)-3-methyl-N-(...)
Affinity DataIC50:  5.70E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305971((S)-N-(4-tert-butylthiazol-2-yl)-2-(4-chlorophenyl...)
Affinity DataIC50:  7.90E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305932(1-(4-chlorophenyl)-N-(5-fluorothiazol-2-yl)cyclohe...)
Affinity DataIC50:  8.50E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305924((S)-2-(4-chlorophenyl)-3-cyclopropyl-N-(thiazol-2-...)
Affinity DataIC50:  8.80E+3nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305943((S)-2-(4-chlorophenyl)-N,3-dimethylbutanamide | CH...)
Affinity DataIC50:  1.10E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305956((S)-2-(4-chlorophenyl)-3-methyl-N-(1,3,4-thiadiazo...)
Affinity DataIC50:  1.20E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305935((S)-2-(2-chloropyridin-4-yl)-2-cyclopropyl-N-(5-fl...)
Affinity DataIC50:  1.60E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305970((S)-2-(4-chlorophenyl)-3-methyl-N-(4-(trifluoromet...)
Affinity DataIC50:  1.70E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50305965((S)-2-(4-chlorophenyl)-3-methyl-N-(4-oxo-4,5-dihyd...)
Affinity DataIC50:  2.00E+4nMAssay Description:Agonist activity at human FFA2 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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