Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50039108
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50423773BDBM50423773(A-1544750 | CEP-701 | KT-5555 | SP924 | LESTAURTIN...)
Affinity DataIC50: 5nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313606BDBM50313606(Sodium-3-[hydroxyimino]-2'-oxo-1,3,1',2'-tetrahydr...)
Affinity DataIC50: 9nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 15nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313610BDBM50313610(5'-Methyl-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 28nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7393BDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataIC50: 33nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304109BDBM50304109(5'-Nitro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3-...)
Affinity DataIC50: 62nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313609BDBM50313609(5'-Chloro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 82nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304112BDBM50304112((Z)-5'-Amino-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 128nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313614BDBM50313614(5'-Methyl-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 209nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313613BDBM50313613(5'-Chloro-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 212nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313615BDBM50313615(Sodium-3,2'-dioxo-1,3,1',2'-tetrahydro-[2,3']biind...)
Affinity DataIC50: 280nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304110BDBM50304110((Z)-5'-Amino-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 359nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7492BDBM7492(3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2...)
Affinity DataIC50: 418nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313608BDBM50313608(5',7'-Dimethyl-1H,1'H-[2,3']biindolylidene-3,2'-di...)
Affinity DataIC50: 952nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of Aurora A by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313612BDBM50313612(5'-Iodo-1H,1'H-[2,3']biindolylidene-3,2'-dione | C...)
Affinity DataIC50: 4.72E+3nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of insulin receptor by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313611BDBM50313611(5'-Trifluoromethoxy-1H,1'H-[2,3']biindolylidene-3,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFR by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Ron by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313604BDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Met by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304121BDBM50304121((Z)-5-Bromo-5'-nitro-1H,1'H-[2,3']biindolylidene-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50304116BDBM50304116((Z)-5'-Nitro-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313607BDBM50313607(5'-Chloro-7'-methyl-1H,1'H-[2,3']biindolylidene-3,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313617BDBM50313617(1-Acetyl-1H,1'H-[2,3']biindolylidene-3,2'-dione | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349806BDBM50349806(INDIRUBIN)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50313616BDBM50313616(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed