Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50031984
TargetAcetylcholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322767(2-Methyl-7-{[8-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322768(5-Chloro-7-{[9-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322767(2-Methyl-7-{[8-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  2nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322766(7-{[9-(1,2,3,4-Tetrahydroacridin-9-ylamino)nonylam...)
Affinity DataIC50:  5nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322766(7-{[9-(1,2,3,4-Tetrahydroacridin-9-ylamino)nonylam...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322768(5-Chloro-7-{[9-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322767(2-Methyl-7-{[8-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of human serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322777(2-Methyl-7-{[10-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  7nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  10nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322766(7-{[9-(1,2,3,4-Tetrahydroacridin-9-ylamino)nonylam...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322766(7-{[9-(1,2,3,4-Tetrahydroacridin-9-ylamino)nonylam...)
Affinity DataIC50:  20nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322770(7-{[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyla...)
Affinity DataIC50:  25nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322782(5-Chloro-7-{{3-{methyl[3-(1,2,3,4-tetrahydroacridi...)
Affinity DataIC50:  30nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322771(7-{[8-(1,2,3,4-Tetrahydroacridin-9-ylamino)octylam...)
Affinity DataIC50:  30nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322772(7-{[10-(1,2,3,4-Tetrahydroacridin-9-ylamino)decyla...)
Affinity DataIC50:  50nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322774(7-{{3-{Methyl[3-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  50nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322768(5-Chloro-7-{[9-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  55nMAssay Description:Inhibition of human serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322772(7-{[10-(1,2,3,4-Tetrahydroacridin-9-ylamino)decyla...)
Affinity DataIC50:  65nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322777(2-Methyl-7-{[10-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  70nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322767(2-Methyl-7-{[8-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  75nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322774(7-{{3-{Methyl[3-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  80nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322768(5-Chloro-7-{[9-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  85nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322771(7-{[8-(1,2,3,4-Tetrahydroacridin-9-ylamino)octylam...)
Affinity DataIC50:  90nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322782(5-Chloro-7-{{3-{methyl[3-(1,2,3,4-tetrahydroacridi...)
Affinity DataIC50:  90nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM32203(8-quinolinol | CHEMBL310555 | US10005735, Table 1....)
Affinity DataIC50: >100nMAssay Description:Inhibition of human serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322776(2-Methyl-7-{[9-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  100nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322780(5-Chloro-7-{[10-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  100nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM32203(8-quinolinol | CHEMBL310555 | US10005735, Table 1....)
Affinity DataIC50: >100nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322770(7-{[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyla...)
Affinity DataIC50:  150nMAssay Description:Inhibition of horse serum BChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322779(5-Chloro-7-{[8-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  150nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322769(7-{[6-(1,2,3,4-Tetrahydroacridin-9-ylamino)hexylam...)
Affinity DataIC50:  200nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322778(2-Methyl-7-{{3-{methyl[3-(1,2,3,4-tetrahydroacridi...)
Affinity DataIC50:  200nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322775(2-Methyl-7-{[7-(1,2,3,4-tetrahydroacridin-9-ylamin...)
Affinity DataIC50:  200nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322773(7-{[12-(1,2,3,4-Tetrahydroacridin-9-ylamino)dodecy...)
Affinity DataIC50:  250nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Bos taurus (bovine))
Instituto De Quimica Medica

Curated by ChEMBL
LigandPNGBDBM50322781(5-Chloro-7-{[12-(1,2,3,4-tetrahydroacridin-9-ylami...)
Affinity DataIC50:  400nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed