Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50039220
TargetZinc finger protein GLI1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50321859(2-(3-Benzoylphenyl)-N-(1H-indol-5-yl)-N-propylprop...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human Gli1 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc finger protein GLI1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50321858(2-(3-Benzoylphenyl)-N-(1H-indol-6-yl)-N-propylprop...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human Gli1 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc finger protein GLI2(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50321859(2-(3-Benzoylphenyl)-N-(1H-indol-5-yl)-N-propylprop...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human Gli2 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc finger protein GLI2(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50321858(2-(3-Benzoylphenyl)-N-(1H-indol-6-yl)-N-propylprop...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human Gli2 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc finger protein GLI1(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50249557(2,2'-(2-(pyridin-4-yl)dihydropyrimidine-1,3(2H,4H)...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human Gli1-mediated transcriptional activity in human Rh30 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed