Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50032337
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50247053BDBM50247053(Tiprolisant | 1-(3-(3-(4-chlorophenyl)propoxy)prop...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327232BDBM50327232(4,5-diphenyl-2-(3-(piperidin-1-yl)propoxy)thiazole...)
Affinity DataKi:  11.2nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327314BDBM50327314(5-ethyl-2-(3-(piperidin-1-yl)propoxy)-4,5,6,7-tetr...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327316BDBM50327316(2-(3-(piperidin-1-yl)propoxy)-5-(3-(piperidin-1-yl...)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327313BDBM50327313(5-methyl-2-(3-(piperidin-1-yl)propoxy)-4,5,6,7-tet...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327320BDBM50327320(4-methyl-5-phenyl-2-(3-(piperidin-1-yl)propoxy)thi...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327319BDBM50327319(4-bromo-5-phenyl-2-(3-(piperidin-1-yl)propoxy)thia...)
Affinity DataKi:  93nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327312BDBM50327312(2-(3-(dimethylamino)propoxy)-6,7-dihydrobenzo[d]th...)
Affinity DataKi:  153nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327321BDBM50327321(1-(5-methyl-2-(3-(piperidin-1-yl)propoxy)thiazol-4...)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327309BDBM50327309(N,N-dimethyl-3-(5-methyl-4,5,6,7-tetrahydrothiazol...)
Affinity DataKi:  257nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327315BDBM50327315(5-benzyl-2-(3-(piperidin-1-yl)propoxy)-4,5,6,7-tet...)
Affinity DataKi:  261nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327318BDBM50327318(2-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-4H-pyran...)
Affinity DataKi:  344nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327317BDBM50327317(2-(3-(piperidin-1-yl)propoxy)-4,5,6,7-tetrahydrobe...)
Affinity DataKi:  357nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327310BDBM50327310(N,N-dimethyl-3-(4,5,6,7-tetrahydrobenzo[d]thiazol-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327311BDBM50327311(3-(6,7-dihydro-4H-pyrano[3,4-d]thiazol-2-yloxy)-N,...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50327322BDBM50327322(2-(3-(piperidin-1-yl)propoxy)-6,7-dihydrobenzo[d]t...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed