BindingDB PrimarySearch

Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50039381

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM50336825((1S,3S,9aS)-1-benzyl-6-((S)-2-(methylamino)propana...)

Kd: 31nMAssay Description:Inhibition of XIAP by FP assayMore data for this Ligand-Target Pair

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM17347((3R,6S,9aR)-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-...)

Ki: 270nMAssay Description:Inhibition of XIAP by FP assayMore data for this Ligand-Target Pair

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM50336824((S)-N-((S)-1-cyclohexyl-2-oxo-2-((3aS,7aR)-5-phene...)

IC50: 280nMAssay Description:Inhibition of XIAP by FRET assayMore data for this Ligand-Target Pair

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM13190((2S)-2-amino-N-[4-(4-bromophenyl)-5-phenyl-1,3-thi...)

Kd: 750nMAssay Description:Inhibition of XIAP by FP assayMore data for this Ligand-Target Pair

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM50336823(1-((S)-2-((S)-2-Aminopropanamido)-3-methylbutanoyl...)

Kd: 2.16E+4nMAssay Description:Inhibition of XIAP-Bir3 domain by calorimetric titration assayMore data for this Ligand-Target Pair

E3 ubiquitin-protein ligase XIAP(Human)
University of Pittsburgh

Curated by ChEMBL

BDBM50336823(1-((S)-2-((S)-2-Aminopropanamido)-3-methylbutanoyl...)

Kd: 2.77E+4nMAssay Description:Inhibition of XIAP-Bir3 domain by NMR titrationMore data for this Ligand-Target Pair