Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50033025
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338329(CHEMBL1681798 | N-(2-{3-[(5-Chlorothiophen-2-yl)ca...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338345(CHEMBL1682882 | N-{2-[4-(3-Oxomorpholin-4-yl)benzo...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338346(CHEMBL1682883 | N-{2-[4-(3-Oxomorpholin-4-yl)pheny...)
Affinity DataIC50:  9nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338336(CHEMBL1682740 | N-[2-({[(5-Chlorothiophen-2-yl)car...)
Affinity DataIC50:  11nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338335(CHEMBL1682739 | N-[3-({[(5-Chlorothiophen-2-yl)car...)
Affinity DataIC50:  12nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338334(CHEMBL1682738 | N-[4-({[(5-Chlorothiophen-2-yl)car...)
Affinity DataIC50:  13nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338333(CHEMBL1682737 | N-[3-({[(5-Chlorothiophen-2-yl)car...)
Affinity DataIC50:  18nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338332(CHEMBL1682736 | N-[(1R*,2R*)-2-({[(5-Chlorothiophe...)
Affinity DataIC50:  27nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338341(CHEMBL1682745 | N-[2-({[(4-Chloro-1H-pyrrol-2-yl)c...)
Affinity DataIC50:  48nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338344(CHEMBL1682881 | N-[2-(5-Methyl-4,5,6,7-tetrahydro[...)
Affinity DataIC50:  59nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338326(CHEMBL1682731 | N-{3-[(5-Chlorothiophen-2-yl)carbo...)
Affinity DataIC50:  93nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338347(CHEMBL1682884 | N-(2-{[(5-Chlorothiophen-2-yl)carb...)
Affinity DataIC50:  204nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338331(CHEMBL1682735 | N-[(1R*,2S*)-2-({[(5-Chlorothiophe...)
Affinity DataIC50:  439nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338343(CHEMBL1682880 | N-(2-{2-[(5-Chloropyridin-2-yl)ami...)
Affinity DataIC50:  623nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338338(CHEMBL1682742 | N-(2-{[(4-Chlorobenzoyl)amino]meth...)
Affinity DataIC50:  642nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338327(CHEMBL1682732 | N-{1-[(5-Methyl-4,5,6,7-tetrahydro...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338340(CHEMBL1682744 | N-(2-{[(3-Chlorobenzoyl)amino]meth...)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338348(CHEMBL1682885 | N-[2-(1-Isopropylpioeridin-4-ylcar...)
Affinity DataIC50:  1.93E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338337(CHEMBL1682741 | N-[2-({[(5-Chloropyridin-2-yl)carb...)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338339(CHEMBL1682743 | N-(2-{[(4-Chloropyridine-2-yl)carb...)
Affinity DataIC50:  4.15E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338330(CHEMBL1682734 | N-(2-{[(5-Chlorothiophen-2-yl)carb...)
Affinity DataIC50:  5.68E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338328(CHEMBL1682733 | N-({1-[(5-Methyl-4,5,6,7-tetrahydr...)
Affinity DataIC50:  6.83E+3nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50338342(CHEMBL1682746 | N-[2-({[(5-Chloro-1H-pyrrol-2-yl)c...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of factor 10a by S2222 chromogenic substrate assay by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed