Compile Data Set for Download or QSAR
maximum 50k data
Found 62 Enz. Inhib. hit(s) with all data for entry = 50033038
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  1nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  1nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338593(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  3nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338600(CHEMBL1683974 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  9nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338599(CHEMBL1683973 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  11nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338596(CHEMBL1683970 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  13nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338609(CHEMBL1683955 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  17nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338591(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  18nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338594(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  19nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338593(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  19nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338589(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  28nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338587(CHEMBL1683961 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  34nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338600(CHEMBL1683974 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  36nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338598(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  38nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338613(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6-me...)
Affinity DataIC50:  65nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338612(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6-me...)
Affinity DataIC50:  68nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338598(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  70nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338594(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  71nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338596(CHEMBL1683970 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  74nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338591(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  78nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338589(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  81nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338599(CHEMBL1683973 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  95nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338595(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  102nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338592(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  114nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338590(CHEMBL1683964 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  120nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338609(CHEMBL1683955 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  140nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338587(CHEMBL1683961 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  150nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338595(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  156nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338590(CHEMBL1683964 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  190nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338588(CHEMBL1683962 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  240nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  240nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338601(5-(4-(benzylamino)but-1-ynyl)-N-(3-chloro-4-(3-flu...)
Affinity DataIC50:  270nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338592(3-(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6...)
Affinity DataIC50:  318nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338588(CHEMBL1683962 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  440nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338614(CHEMBL1683960 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  590nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338610(CHEMBL1683956 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  640nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338612(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6-me...)
Affinity DataIC50:  740nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  760nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338601(5-(4-(benzylamino)but-1-ynyl)-N-(3-chloro-4-(3-flu...)
Affinity DataIC50:  810nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50182914(CHEMBL205652 | N-(4-(3-fluorobenzyloxy)-3-chloroph...)
Affinity DataIC50:  920nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338603(CHEMBL1683949 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338604(CHEMBL1683950 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338613(4-(3-chloro-4-(3-fluorobenzyloxy)phenylamino)-6-me...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338610(CHEMBL1683956 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338614(CHEMBL1683960 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  3.75E+3nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338597(CHEMBL1683971 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  4.13E+3nMAssay Description:Inhibition of EGFR by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338597(CHEMBL1683971 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  5.38E+3nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50338604(CHEMBL1683950 | N-(3-chloro-4-(3-fluorobenzyloxy)p...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of HER2 by homogeneous time-resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 62 total ) | Next | Last >>
Jump to: