Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50004556
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 3nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484055(CHEMBL1808163)
Affinity DataIC50: 18nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484048(CHEMBL1808162)
Affinity DataIC50: 22nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484049(CHEMBL1808165)
Affinity DataIC50: 54nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484056(CHEMBL1807694)
Affinity DataIC50: 55nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484046(CHEMBL1807693)
Affinity DataIC50: 62nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 67nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484060(CHEMBL1808168)
Affinity DataIC50: 77nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484058(CHEMBL1808167)
Affinity DataIC50: 90nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484057(CHEMBL1808173)
Affinity DataIC50: 94nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484052(CHEMBL1808172)
Affinity DataIC50: 111nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484054(CHEMBL1808166)
Affinity DataIC50: 115nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484061(CHEMBL1808160)
Affinity DataIC50: 132nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484047(CHEMBL1808161)
Affinity DataIC50: 137nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484050(CHEMBL1808169)
Affinity DataIC50: 171nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484051(CHEMBL1808170)
Affinity DataIC50: 403nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484059(CHEMBL1808171)
Affinity DataIC50: 510nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50484053(CHEMBL1808164)
Affinity DataIC50: 838nMAssay Description:Inhibition of HDAC in human HeLa cells using Ac-Arg-Gly-Lys(Ac)-AMC as fluorescent substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed