Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50039422
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347177BDBM50347177(CHEMBL1797687)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347179BDBM50347179(CHEMBL1797689)
Affinity DataKi:  0.0380nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347179BDBM50347179(CHEMBL1797689)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347178BDBM50347178(CHEMBL1797688)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347177BDBM50347177(CHEMBL1797687)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347178BDBM50347178(CHEMBL1797688)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001707BDBM50001707(Tylox | Oxycet | Combunox | Codoxy | Percocet | 10...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000092BDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347175BDBM50347175(CHEMBL1797685)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347174BDBM50347174(CHEMBL1797684)
Affinity DataKi:  17.4nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347176BDBM50347176(CHEMBL1797686)
Affinity DataKi:  21.7nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000092BDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  46.9nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001707BDBM50001707(Tylox | Oxycet | Combunox | Codoxy | Percocet | 10...)
Affinity DataKi:  57.6nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347174BDBM50347174(CHEMBL1797684)
Affinity DataKi:  58.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347176BDBM50347176(CHEMBL1797686)
Affinity DataKi:  77.7nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrain homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347175BDBM50347175(CHEMBL1797685)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/8/2013
Entry Details Article
PubMed