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Found 93 Enz. Inhib. hit(s) with all data for entry = 50039482
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50366495((+)butaclamol | CHEMBL1255588)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354102(CHEMBL1836107)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM31005(2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyraz...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354098(CHEMBL1836061)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354103(CHEMBL1836108)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354104(CHEMBL1836109)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354100(CHEMBL1836105)
Affinity DataKi:  12.3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354115(CHEMBL1836054)
Affinity DataKi:  16.6nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354115(CHEMBL1836054)
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354114(CHEMBL1836056)
Affinity DataKi:  24.1nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354091(CHEMBL1836044)
Affinity DataKi:  26.3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354105(CHEMBL1836110)
Affinity DataKi:  28.3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354102(CHEMBL1836107)
Affinity DataKi:  82.4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354098(CHEMBL1836061)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354096(CHEMBL1836059)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354111(CHEMBL1836052)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354109(CHEMBL1836050)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354114(CHEMBL1836056)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354109(CHEMBL1836050)
Affinity DataKi:  218nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50095890(2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperaz...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354102(CHEMBL1836107)
Affinity DataKi:  304nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354101(CHEMBL1836106)
Affinity DataKi:  394nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354099(CHEMBL1836104)
Affinity DataKi:  394nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354110(CHEMBL1836051)
Affinity DataKi:  507nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354101(CHEMBL1836106)
Affinity DataKi:  532nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354092(CHEMBL1836045)
Affinity DataKi:  653nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354111(CHEMBL1836052)
Affinity DataKi:  682nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354105(CHEMBL1836110)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354091(CHEMBL1836044)
Affinity DataKi:  745nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354107(CHEMBL1836048 | cid_653771)
Affinity DataKi:  929nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354104(CHEMBL1836109)
Affinity DataKi:  956nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354103(CHEMBL1836108)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354090(CHEMBL1836043)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354093(CHEMBL1836046)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354108(CHEMBL1836049)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354095(CHEMBL1836058)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354093(CHEMBL1836046)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354097(CHEMBL1836060)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354100(CHEMBL1836105)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354092(CHEMBL1836045)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354103(CHEMBL1836108)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354110(CHEMBL1836051)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354111(CHEMBL1836052)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354113(CHEMBL1836055)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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