Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50033961
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354637(CHEMBL1834440)
Affinity DataIC50: 14nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354642(CHEMBL1834204)
Affinity DataIC50: 14nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354639(CHEMBL1834201)
Affinity DataIC50: 17nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354638(CHEMBL1834200)
Affinity DataIC50: 18nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM20716((1R,2R)-2-[(4-{4-[(phenylcarbamoyl)amino]phenyl}ph...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human DGAT1 expressed in Sf9 cells assessed as formation of didecanoylglycerol product after 1 hr using 14C-decanoyl-CoA by beta scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM20716((1R,2R)-2-[(4-{4-[(phenylcarbamoyl)amino]phenyl}ph...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354641(CHEMBL1834203)
Affinity DataIC50: 25nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354631(CHEMBL1834433)
Affinity DataIC50: 28nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354629(CHEMBL1834431)
Affinity DataIC50: 30nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354634(CHEMBL1834436)
Affinity DataIC50: 32nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354633(CHEMBL1834435)
Affinity DataIC50: 51nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354636(CHEMBL1834438)
Affinity DataIC50: 57nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354640(CHEMBL1834202)
Affinity DataIC50: 64nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354630(CHEMBL1834432)
Affinity DataIC50: 72nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354643(CHEMBL1834206)
Affinity DataIC50: 73nMAssay Description:Inhibition of human DGAT1 expressed in Sf9 cells assessed as formation of didecanoylglycerol product after 1 hr using 14C-decanoyl-CoA by beta scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354632(CHEMBL1834434)
Affinity DataIC50: 88nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDiacylglycerol O-acyltransferase 1(Human)
Piramal Life Sciences

Curated by ChEMBL
LigandPNGBDBM50354635(CHEMBL1834437)
Affinity DataIC50: 99nMAssay Description:Inhibition of human DGAT1 assessed as formation of [14C]-triglyceride using [14C]oleoyl-CoA by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed