Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50033977
TargetCannabinoid receptor 1(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354843(BAY-387271 | CHEMBL1668508)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to recombinant human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  45.5nMAssay Description:Displacement of [3H]BAY-38-7271 from recombinant human CB2 receptor expressed in CHO cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  45.5nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  48.3nMAssay Description:Displacement of [3H]BAY-38-7271 from CB1 receptor in human brain cortex membranes after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  55.4nMAssay Description:Displacement of [3H]BAY-38-7271 from CB1 receptor in Wistar rat brain membranes after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM86514(BAY 59-3074 | CAS_406205-74-1 | CHEMBL1354658)
Affinity DataKi:  55.4nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354847(CHEMBL1834525)
Affinity DataKi:  253nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354846(CHEMBL1834524)
Affinity DataKi:  317nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354846(CHEMBL1834524)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]CP55940 from mouse cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354847(CHEMBL1834525)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]CP55940 from mouse cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354844(CHEMBL1834522)
Affinity DataKi:  676nMAssay Description:Displacement of [3H]CP55940 from mouse cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354846(CHEMBL1834524)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354848(CHEMBL1834526)
Affinity DataKi:  1.13E+3nMAssay Description:Displacement of [3H]CP55940 from mouse cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354848(CHEMBL1834526)
Affinity DataKi:  1.16E+3nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354845(CHEMBL1834523)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]CP55940 from mouse cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354844(CHEMBL1834522)
Affinity DataKi:  1.81E+3nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354844(CHEMBL1834522)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354847(CHEMBL1834525)
Affinity DataKi:  2.28E+3nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354845(CHEMBL1834523)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354845(CHEMBL1834523)
Affinity DataKi:  3.29E+3nMAssay Description:Displacement of [3H]CP55940 from human cannabinoid CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50354848(CHEMBL1834526)
Affinity DataKi:  1.44E+4nMAssay Description:Displacement of [3H]CP55940 from rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed