Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 8344
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 20nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM50022775(m-Trimethylammoniumphenyldimethylcarbamate | Prost...)
Affinity DataIC50: 50nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241985(4-[5-(2,4-Dichlorophenoxymethyl)-1,3,4-thiadiazol-...)
Affinity DataIC50: 53nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241978(4-(5-Heptyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol...)
Affinity DataIC50: 60nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM50022775(m-Trimethylammoniumphenyldimethylcarbamate | Prost...)
Affinity DataIC50: 70nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241983(4-(5-{4-[5-(2,4-Dihydroxyphenyl)-1,3,4-thiadiazol-...)
Affinity DataIC50: 92nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241990(4-Chloro-6-(5-(4-fluorophenylamino)-1,3,4-thiadiaz...)
Affinity DataIC50: 105nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241977(4-(5-Propyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol...)
Affinity DataIC50: 109nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241988(4-{5-[5-(4-Bromophenyl)thiophen-2-yl]-1,3,4-thiadi...)
Affinity DataIC50: 125nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241990(4-Chloro-6-(5-(4-fluorophenylamino)-1,3,4-thiadiaz...)
Affinity DataIC50: 143nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241981(4,4'-[5,5'-Methylenedi-(1,3,4-thiadiazole-...)
Affinity DataIC50: 184nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241980(4-[5-(1,3-Benzodioxol-5-yl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 220nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241978(4-(5-Heptyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol...)
Affinity DataIC50: 240nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241981(4,4'-[5,5'-Methylenedi-(1,3,4-thiadiazole-...)
Affinity DataIC50: 260nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241992(4-Chloro-6-(5-(3,4-dihydroxyphenyl)-1,3,4-thiadiaz...)
Affinity DataIC50: 1.27E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241984(4-(5-(4-(Trifluoromethyl)phenylamino)-1,3,4-thiadi...)
Affinity DataIC50: 1.32E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241991(4-Chloro-6-(5-(3-chlorophenylamino)-1,3,4-thiadiaz...)
Affinity DataIC50: 2.68E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241982(4,4'-{[5,5'-(Ethane-1,2-diyl)]di(1,3,4-thi...)
Affinity DataIC50: 3.11E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241984(4-(5-(4-(Trifluoromethyl)phenylamino)-1,3,4-thiadi...)
Affinity DataIC50: 3.24E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 7.52E+3nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241982(4,4'-{[5,5'-(Ethane-1,2-diyl)]di(1,3,4-thi...)
Affinity DataIC50: 1.43E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241983(4-(5-{4-[5-(2,4-Dihydroxyphenyl)-1,3,4-thiadiazol-...)
Affinity DataIC50: 1.52E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241989(4-(5-Benzyl-1,3,4-thiadiazol-2-yl)-6-chlorobenzene...)
Affinity DataIC50: 1.80E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241977(4-(5-Propyl-1,3,4-thiadiazol-2-yl)benzene-1,3-diol...)
Affinity DataIC50: 1.82E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241988(4-{5-[5-(4-Bromophenyl)thiophen-2-yl]-1,3,4-thiadi...)
Affinity DataIC50: 1.86E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241980(4-[5-(1,3-Benzodioxol-5-yl)-1,3,4-thiadiazol-2-yl]...)
Affinity DataIC50: 2.51E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241992(4-Chloro-6-(5-(3,4-dihydroxyphenyl)-1,3,4-thiadiaz...)
Affinity DataIC50: 3.52E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241987(4-{5-[5-(4-Fluorophenyl)thiophen-2-yl]-1,3,4-thiad...)
Affinity DataIC50: 3.72E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241989(4-(5-Benzyl-1,3,4-thiadiazol-2-yl)-6-chlorobenzene...)
Affinity DataIC50: 4.42E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241986(4-{5-[5-(4-Bromophenyl)-1,2-oxazol-3-yl]-1,3,4-thi...)
Affinity DataIC50: 4.52E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241985(4-[5-(2,4-Dichlorophenoxymethyl)-1,3,4-thiadiazol-...)
Affinity DataIC50: 5.02E+4nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241986(4-{5-[5-(4-Bromophenyl)-1,2-oxazol-3-yl]-1,3,4-thi...)
Affinity DataIC50: 1.93E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241979(4-[5-(Naphthalen-2-yl)-1,3,4-thiadiazol-2-yl]benze...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241979(4-[5-(Naphthalen-2-yl)-1,3,4-thiadiazol-2-yl]benze...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241993(3-{5-[4-(Dimethylamino)phenyl]-1,3,4-thiadiazol-2-...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Life Sciences

LigandPNGBDBM241993(3-{5-[4-(Dimethylamino)phenyl]-1,3,4-thiadiazol-2-...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241991(4-Chloro-6-(5-(3-chlorophenylamino)-1,3,4-thiadiaz...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Horse)
University of Life Sciences

LigandPNGBDBM241987(4-{5-[5-(4-Fluorophenyl)thiophen-2-yl]-1,3,4-thiad...)
Affinity DataIC50: 5.00E+5nMpH: 8.0 T: 2°CAssay Description:Seven different concentrations of the synthesized compounds in the range 10^−3-10^−9 M were measured at 412 nm. All the assays were under...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details Article
PubMed